SCHEMBL10344387

SCHEMBL10344387

CCOC(=O)CCCOc1ccc2c(c1)OC(C)(CCCCI)CC2=O

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.49
KDM4E B2RXH2 6/20 0.47
ALDH1A1 P00352 6/20 0.47
HPGD P15428 4/20 0.47
GAA P10253 4/20 0.47
CASP1 P29466 3/20 0.47
HSD17B10 Q99714 3/20 0.47
PDK2 Q15119 2/20 0.43
MAOB P27338 6/20 0.42
PDE3B Q13370 2/20 0.41
PDE3A Q14432 2/20 0.41
P2RY12 Q9H244 1/20 0.41
NPC1 O15118 1/20 0.41
MAPK1 P28482 1/20 0.41
RAB9A P51151 1/20 0.41
GLA P06280 1/20 0.40
ALDH2 P05091 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10695261 0.92 BRD4 (0.50) BRD4KDM4EALDH1A1HPGDGAA
SCHEMBL10704709 0.83 MEN1 (0.43) BRD4KDM4EALDH1A1HPGDGAA
SCHEMBL10694125 0.83 KDM4E (0.47) KDM4EALDH1A1HPGDGAACASP1
SCHEMBL10689874 0.80 CYSLTR1 (0.49)
SCHEMBL10344312 0.80 MAOB (0.46) KDM4EALDH1A1HPGDGAACASP1
SCHEMBL10692495 0.79 LTB4R (0.44) BRD4KDM4EALDH1A1HPGDGAA
SCHEMBL9635631 0.76 KDM4E (0.54) KDM4EALDH1A1HPGDGAACASP1
SCHEMBL9512184 0.76 KDM4E (0.46) BRD4KDM4EALDH1A1HPGDGAA
SCHEMBL10691900 0.74 ALDH1A1 (0.48) KDM4EALDH1A1HPGDGAACASP1
SCHEMBL22578031 0.74 BRD4 (0.65) BRD4ALDH1A1HPGDMAOBNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0261254-B1 3,4-DIHYDRO-4-OXO-2H-1-BENZOPYRANYLOXY ALKANOIC ACID DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1990-02-07 EP disclosed
EP-0261254-A1 3,4-Dihydro-4-oxo-2H-1-benzopyranyloxy alkanoic acid derivatives F. HOFFMANN-LA ROCHE AG (CH) 1988-03-30 EP disclosed
US-4650812-A ANTIALLERGY HOFFMANN-LA ROCHE INC. (US) 1987-03-17 US disclosed