SCHEMBL9511770

SCHEMBL9511770

CCCc1c(O)ccc2c1OC(CCC(=O)OC)(CCC(=O)N1CCCC1)CC2=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.35
HPGD P15428 4/20 0.35
KDM4E B2RXH2 3/20 0.35
GAA P10253 3/20 0.35
GLA P06280 3/20 0.35
NPC1 O15118 2/20 0.35
SMN1; SMN2 Q16637 3/20 0.33
HIF1A Q16665 1/20 0.32
RAB9A P51151 1/20 0.32
MAPT P10636 1/20 0.32
POLB P06746 1/20 0.32
ADAMTS5 Q9UNA0 1/20 0.32
LTB4R Q15722 1/20 0.31
LTB4R2 Q9NPC1 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
CASP3 P42574 1/20 0.31
CASP2 P42575 1/20 0.31
CASP7 P55210 1/20 0.31
CASP6 P55212 1/20 0.31
CASP8 Q14790 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9511722 0.91 LTB4R (0.35) ALDH1A1HPGDKDM4EGAAGLA
SCHEMBL10374275 0.85 AKT1 (0.38) ALDH1A1HPGDKDM4EGAAGLA
SCHEMBL9485831 0.83 ALDH1A1 (0.36) ALDH1A1HPGDKDM4EGAAGLA
SCHEMBL9821761 0.81 AKT1 (0.38) ALDH1A1HPGDKDM4EGAASMN1; SMN2
SCHEMBL9512199 0.80 LTB4R (0.39) LTB4RLTB4R2KMT2A
SCHEMBL10368286 0.79 LTB4R (0.33) LTB4RLTB4R2
SCHEMBL9511662 0.74 ESR1 (0.33) ALDH1A1KDM4EGAAMAPTPOLB
SCHEMBL9515500 0.73 LTB4R (0.42) LTB4RLTB4R2
SCHEMBL10371731 0.73 AKT1 (0.39) ALDH1A1HPGDKDM4EGAAGLA
SCHEMBL9511741 0.72 ESR1 (0.32) KDM4EGAAMAPTPOLBLTB4R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0342664-B1 2,2-disubstituted benzopyran leukotriene-D4 antagonists SEARLE & CO (US) 1993-12-15 EP disclosed
US-5093353-A 2,2-di-substituted benzopyran leukotriene-D4 antagonists G. D. SEARLE & CO. (US) 1992-03-03 US disclosed
EP-0342664-A2 2,2-disubstituted benzopyran leukotriene-D4 antagonists G.D. Searle & Co. (US) 1989-11-23 EP disclosed