SCHEMBL9512958

SCHEMBL9512958

COc1cc(OC)cc(C(=O)N2CCN(CCc3ccc(Cl)cc3)CC2)c1

nearest known ligand 0.61

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 3/20 0.60
THRB P10828 1/20 0.60
DRD3 P35462 2/20 0.60
KCNA5 P22460 1/20 0.60
HTR2A P28223 2/20 0.54
ALDH1A1 P00352 3/20 0.53
KDM4E B2RXH2 2/20 0.53
LMNA P02545 1/20 0.53
SIGMAR1 Q99720 1/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
KCNH2 Q12809 1/20 0.52
TSHR P16473 1/20 0.52
HTT P42858 1/20 0.52
WNK1 Q9H4A3 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9513158 0.99 DRD2 (0.59) DRD2THRBDRD3KCNA5HTR2A
SCHEMBL9513026 0.90 WNK1 (0.64) DRD2THRBDRD3KCNA5ALDH1A1
SCHEMBL9514261 0.89 DRD2 (0.76) DRD2THRBDRD3KCNA5HTR2A
Hydrochloric Acid SCHEMBL9513192 0.89 WNK1 (0.63) DRD2THRBDRD3KCNA5ALDH1A1
SCHEMBL9513265 0.88 THRB (0.58) DRD2THRBDRD3KCNA5HTR2A
Hydrochloric Acid SCHEMBL9514254 0.87 THRB (0.57) DRD2THRBDRD3KCNA5HTR2A
SCHEMBL9515612 0.85 THRB (0.68) THRBDRD3KCNA5HTR2AALDH1A1
SCHEMBL9513235 0.84 KMT2A (0.67) DRD2THRBDRD3KCNA5ALDH1A1
Hydrochloric Acid SCHEMBL9516717 0.84 THRB (0.67) THRBDRD3KCNA5HTR2AALDH1A1
SCHEMBL9513241 0.83 THRB (0.82) DRD2THRBDRD3KCNA5HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0250361-B1 Disubstituted piperazines CIBA GEIGY AG (CH) 1993-12-08 EP claimed
US-4804661-A ANALGESICS CIBA-GEIGY CORPORATION (US) 1989-02-14 US claimed
EP-0250361-A2 Disubstituted piperazines CIBA-GEIGY AG (CH) 1987-12-23 EP claimed
EP-0250361-B1 Disubstituted piperazines CIBA GEIGY AG (CH) 1993-12-08 EP disclosed
US-4804661-A ANALGESICS CIBA-GEIGY CORPORATION (US) 1989-02-14 US disclosed
EP-0250361-A2 Disubstituted piperazines CIBA-GEIGY AG (CH) 1987-12-23 EP disclosed