SCHEMBL9514683

SCHEMBL9514683

Cc1cc(C)c(C(C)Br)c(C)c1

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
RAPGEF4 Q8WZA2 4/20 0.38
SLC6A2 P23975 2/20 0.35
SLC6A4 P31645 2/20 0.35
SLC6A3 Q01959 2/20 0.35
ALDH1A1 P00352 2/20 0.32
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP2A6 P11509 1/20 0.31
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28231414 0.79 CYP3A4 (0.44) ALDH1A1GAA
SCHEMBL8053821 0.78 RAPGEF4 (0.38) RAPGEF4SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL5163137 0.77 RAPGEF4 (0.41) RAPGEF4SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL27927634 0.77 RAPGEF4 (0.41) RAPGEF4SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL10832009 0.76 LMNA (0.31) RAPGEF4LMNA
SCHEMBL28231322 0.75 ALDH1A1 (0.43) ALDH1A1GAATSHR
SCHEMBL18243433 0.74 RAPGEF4 (0.35) RAPGEF4SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL8732505 0.74 NR3C1 (0.36) RAPGEF4SLC6A2SLC6A4SLC6A3TSHR
SCHEMBL2848311 0.73 RAPGEF4 (0.43) RAPGEF4SLC6A2SLC6A4SLC6A3ALDH1A1
SCHEMBL23122285 0.72 RAPGEF4 (0.38) RAPGEF4SLC6A2SLC6A4SLC6A3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0454270-B1 Catalyst compositions SHELL INT RESEARCH (NL) 1993-12-15 EP claimed
CN-108503579-B Fentanyl analogs and uses thereof 南京医科大学 2021-03-26 CN disclosed
CN-108503579-A Fentanyl analog and its application 南京医科大学 2018-09-07 CN disclosed
CN-101671240-B Method for preparing 2,2-dimethyl-3-hydrocinnnamic aldehyde and derivative thereof SHANGHAI INST TECHNOLOGY 2013-06-19 CN disclosed