SCHEMBL9516545

SCHEMBL9516545

COc1ccc(C2=C(C=O)c3ccc(OC)cc3CC2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MIF P14174 4/20 0.45
ESR1 P03372 1/20 0.43
CYP19A1 P11511 3/20 0.43
ALDH1A1 P00352 3/20 0.43
MAPT P10636 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
CYP26A1 O43174 3/20 0.43
LMNA P02545 1/20 0.43
CYP11B2 P19099 2/20 0.43
EBP Q15125 1/20 0.42
SIGMAR1 Q99720 1/20 0.42
MAPK1 P28482 1/20 0.42
EGFR P00533 1/20 0.42
KDM4E B2RXH2 2/20 0.42
GLA P06280 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP27A1 Q02318 1/20 0.41
NPC1 O15118 1/20 0.41
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3654013 0.78 ESR1 (0.53) ESR1CYP19A1CYP11B2EBPSIGMAR1
SCHEMBL10470879 0.77 MIF (0.48) MIFESR1CYP19A1ALDH1A1MAPT
SCHEMBL3141978 0.76 MPO (0.54) MIFCYP19A1ALDH1A1MAPTSMN1; SMN2
SCHEMBL7628081 0.76 ESR1 (0.63) MIFESR1ALDH1A1MAPTSMN1; SMN2
SCHEMBL28448661 0.75 ESR2 (0.47) MIFESR1CYP26A1
SCHEMBL9516552 0.74 EGFR (0.50) ESR1CYP19A1ALDH1A1MAPTLMNA
SCHEMBL9516797 0.74 KDM4E (0.47) MIFESR1CYP19A1ALDH1A1MAPT
SCHEMBL3862097 0.74 ESR1 (0.52) ESR1ALDH1A1MAPTSMN1; SMN2KDM4E
SCHEMBL17108416 0.74 MPO (0.59) MIFCYP19A1ALDH1A1MAPTSMN1; SMN2
SCHEMBL7623247 0.73 ESR1 (0.75) MIFESR1CYP26A1EBPSIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0394194-B1 PROTECTED AMINO-ACIDS AND PROCESS FOR THEIR PREPARATION CALBIOCHEM-NOVABIOCHEM AG (CH) 1993-08-18 EP claimed
CN-107406424-B Estrogen receptor modulators and uses thereof 豪夫迈·罗氏有限公司 2020-08-25 CN disclosed
EP-0281283-B1 HETEROCYCLIC COMPOUNDS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-02-10 EP disclosed
US-4910212-A Containing 1,2,4-triazole or imidazole ring IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-03-20 US disclosed
EP-0281283-A1 Heterocyclic compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1988-09-07 EP disclosed