SCHEMBL9517099

SCHEMBL9517099

Cc1ccc(NS(=O)(=O)c2cccc(C(F)(F)F)c2)cn1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.69
HSD17B2 P37059 1/20 0.62
KMT2A Q03164 4/20 0.58
SLC22A12 Q96S37 1/20 0.58
NR3C1 P04150 1/20 0.57
PGR P06401 1/20 0.57
AR P10275 1/20 0.57
ESR2 Q92731 1/20 0.57
PIK3CB P42338 1/20 0.56
FFAR1 O14842 1/20 0.55
CDK1 P06493 1/20 0.55
CCNB1 P14635 1/20 0.55
CCNA2 P20248 1/20 0.55
CDK2 P24941 1/20 0.55
CDK7 P50613 1/20 0.55
CCNH P51946 1/20 0.55
CCNA1 P78396 1/20 0.55
FFAR4 Q5NUL3 1/20 0.55
SLC40A1 Q9NP59 1/20 0.55
CLK1 P49759 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9516051 0.88 PSEN1 (0.64) TSHRHSD17B2KMT2ASLC22A12FFAR1
SCHEMBL9517269 0.84 SLC22A12 (0.60) TSHRKMT2ASLC22A12ARFFAR1
SCHEMBL9517147 0.83 PGR (0.54) KMT2ASLC22A12PGRHDAC1HDAC8
SCHEMBL9517143 0.81 TSHR (0.61) TSHRHSD17B2KMT2ANR3C1PGR
SCHEMBL7572806 0.81 NR3C1 (0.69) TSHRHSD17B2KMT2ANR3C1PGR
SCHEMBL7573925 0.80 HSD17B2 (0.79) TSHRHSD17B2KMT2ANR3C1PGR
SCHEMBL97543 0.80 NR3C1 (0.67) TSHRHSD17B2KMT2ANR3C1PGR
SCHEMBL30926704 0.79 GAA (0.57) TSHRHSD17B2KMT2AFFAR1CDK1
SCHEMBL27180634 0.79 GAA (0.57) TSHRHSD17B2KMT2AFFAR1CDK1
SCHEMBL13248888 0.79 HSD17B2 (0.53) TSHRHSD17B2KMT2ANR3C1PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1079466-A 4-or 5-(sulphur) acylimino-and (inferior sulphur) amidopyridine and pyridine-N-oxide thereof HOECHST AG (DE) 1993-12-15 CN disclosed
EP-0567997-A1 4- or 5-(sulf)imido- and (sulfon)amidopyridines and their pyridine-N-oxides, process for their preparation and their use as pharmaceutical HOECHST AKTIENGESELLSCHAFT (DE) 1993-11-03 EP disclosed