SCHEMBL9519154

SCHEMBL9519154

Cc1cnc(C2=CCCNC2)s1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 3/20 0.40
CHRM3 P20309 2/20 0.40
HTR2A P28223 8/20 0.35
HTR2C P28335 3/20 0.35
HTR2B P41595 3/20 0.35
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
CHRM4 P08173 1/20 0.34
CHRM5 P08912 1/20 0.34
CHRM1 P11229 1/20 0.34
NOS1 P29475 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15001490 0.73 HRH3 (0.42) HTR2AHTR2C
SCHEMBL9149638 0.70 HTR2A (0.38) CHRM2CHRM3HTR2AHTR2CHTR2B
SCHEMBL9151997 0.69 ADRA2A (0.37) CHRM2CHRM3HTR2AHTR2CHTR2B
Hydrochloric Acid SCHEMBL9772133 0.69 CHRM2 (0.36) CHRM2CHRM3HTR2AHTR2CHTR2B
SCHEMBL8400415 0.69 CHRM1 (0.48) CHRM2CHRM3CHRM4CHRM5CHRM1
Hydrochloric Acid SCHEMBL9148160 0.69 HTR2A (0.37) CHRM2CHRM3HTR2AHTR2CHTR2B
SCHEMBL10002194 0.69 NOS1 (0.55) NOS1
Hydrochloric Acid SCHEMBL9148120 0.68 ADRA2A (0.36) CHRM2CHRM3HTR2AHTR2CHTR2B
SCHEMBL14510156 0.68 NOS1 (0.34) NOS1
SCHEMBL9154724 0.67 HTR2A (0.35) CHRM2CHRM3HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0296721-B1 HETEROCYCLIC COMPOUNDS H. LUNDBECK A/S (DK) 1993-06-23 EP disclosed
US-4925858-A NERVOUS SYSTEM DISORDERS, ALZHEIMER*S DISEASE H. LUNDBECK A/S (DK) 1990-05-15 US disclosed
US-4866077-A TREATMENT OF NERVOUS SYSTEM DISORDERS SUCH AS ALZHEIMER*S DISEASE H. LUNDBECK A/S (DK) 1989-09-12 US disclosed
EP-0296721-A2 Heterocyclic compounds H. LUNDBECK A/S (DK) 1988-12-28 EP disclosed