SCHEMBL9520586

SCHEMBL9520586

COc1cccc2c1CC(c1ccccc1)CC2=O

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.54
ALDH1A1 P00352 5/20 0.51
KDM4E B2RXH2 4/20 0.51
LMNA P02545 4/20 0.51
MEN1 O00255 1/20 0.51
KMT2A Q03164 1/20 0.51
RAB9A P51151 2/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
HTT P42858 2/20 0.49
HPGD P15428 1/20 0.48
HSD17B10 Q99714 1/20 0.48
CYP19A1 P11511 1/20 0.48
MAP1LC3B Q9GZQ8 1/20 0.45
LDHA P00338 1/20 0.45
ADRA1D P25100 1/20 0.44
ADRA1A P35348 1/20 0.44
ADRA1B P35368 1/20 0.44
MAPT P10636 3/20 0.44
NPC1 O15118 1/20 0.44
POLB P06746 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7313225 0.84 ALDH1A1 (0.55) ACHEALDH1A1KDM4ELMNAMEN1
SCHEMBL9802182 0.82 ALDH1A1 (0.50) ALDH1A1KDM4ELMNAMEN1KMT2A
SCHEMBL1699532 0.79 ACHE (0.63) ACHEALDH1A1KDM4ELMNAHPGD
SCHEMBL14939214 0.78 ACHE (0.62) ACHEALDH1A1KDM4ELMNAHPGD
SCHEMBL6076000 0.75 HTR7 (0.68) ADRA1DADRA1AADRA1B
SCHEMBL6075908 0.74 KMT2A (0.48) ALDH1A1KDM4ELMNAMEN1KMT2A
Hydrochloric Acid SCHEMBL6490470 0.74 HTR7 (0.67) ADRA1DADRA1AADRA1B
SCHEMBL29506042 0.73 KDM4E (0.61) ACHEALDH1A1KDM4ELMNAMEN1
SCHEMBL165220 0.73 KDM4E (0.61) ACHEALDH1A1KDM4ELMNAMEN1
SCHEMBL6075690 0.73 CYP1A2 (0.56) ACHEKDM4ELMNARAB9ACYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0325963-B1 1-AMINOMETHYL-1,2,3,4-TETRAHYDRONAPHTHALENES AND -INDANES ABBOTT LABORATORIES (US) 1993-09-22 EP disclosed
US-5140040-A Alpha-2-adrenergic receptor antagonist; glaucoma; congestive heart failure; hypotensive agents; headaches; metabolic disorders (diabetes, obesity) ABBOTT LABORATORIES (US) 1992-08-18 US disclosed
US-5128362-A Antidepressant, antiglaucoma ABBOTT LABORATORIES (US) 1992-07-07 US disclosed
US-5086074-A Selective adrenergic receptor antagonists ABBOTT LABORATORIES (US) 1992-02-04 US disclosed
US-4994486-A Neurological disorders ABBOTT LABORATORIES (US) 1991-02-19 US disclosed
EP-0395734-A4 1-AMINOMETHYL-1,2,3,4-TETRAHYDRONAPHTHALENES 1991-01-02 EP disclosed
EP-0395734-A1 1-AMINOMETHYL-1,2,3,4-TETRAHYDRONAPHTHALENES ABBOTT LABORATORIES (US) 1990-11-07 EP disclosed
EP-0325963-A1 1-Aminomethyl-1,2,3,4-tetrahydronaphthalenes and -indanes ABBOTT LABORATORIES (US) 1989-08-02 EP disclosed
WO-1989006645-A1 1-AMINOMETHYL-1,2,3,4-TETRAHYDRONAPHTHALENES ABBOTT LABORATORIES (US) 1989-07-27 WO disclosed