SCHEMBL9520705

SCHEMBL9520705

Cc1cc(N)cc(C)c1S(=O)O

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.38
ALDH1A1 P00352 2/20 0.38
TSHR P16473 2/20 0.38
CASP1 P29466 2/20 0.33
TDP1 Q9NUW8 2/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
MAPT P10636 2/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL345129 0.80 CA1 (0.37) ALDH1A1TDP1KDM4EMAPT
SCHEMBL12856118 0.80 CA1 (0.37) ALDH1A1TDP1KDM4EMAPT
SCHEMBL1022571 0.78 CA1 (0.35) ALDH1A1TDP1KDM4EMAPT
SCHEMBL1022384 0.78 CA1 (0.35) ALDH1A1TDP1KDM4EMAPT
SCHEMBL1023387 0.78 CA1 (0.35) ALDH1A1TDP1KDM4EMAPT
SCHEMBL1024671 0.78 CA1 (0.35) ALDH1A1TDP1KDM4EMAPT
SCHEMBL9740926 0.76 NMT1 (0.35) ALDH1A1KDM4EMEN1KMT2AMAPT
SCHEMBL9739995 0.74 NMT1 (0.34) ALDH1A1KDM4EMEN1KMT2ACYP1A2
SCHEMBL16404373 0.74 POLB (0.43) ALDH1A1TSHRTDP1CYP2C19
SCHEMBL6730284 0.71 PGK1 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0408713-B1 PHENYLSULPHONE DERIVATIVES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-05-19 EP claimed
EP-0408713-A1 PHENYLSULPHONE DERIVATIVES. ICI PLC (GB) 1991-01-23 EP claimed
WO-1990008761-A1 PHENYLSULPHONE DERIVATIVES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-08-09 WO claimed
EP-0408713-B1 PHENYLSULPHONE DERIVATIVES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-05-19 EP disclosed
EP-0408713-A1 PHENYLSULPHONE DERIVATIVES. ICI PLC (GB) 1991-01-23 EP disclosed
WO-1990008761-A1 PHENYLSULPHONE DERIVATIVES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-08-09 WO disclosed