SCHEMBL9521056

SCHEMBL9521056

O=C(NCCSC[C@@H]1C[C@H](SC(=O)c2ccccc2)CN1C(=O)OCc1ccc([N+](=O)[O-])cc1)OCc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP8 Q6V1X1 1/20 0.41
DPP9 Q86TI2 1/20 0.41
ATM Q13315 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
TGM2 P21980 1/20 0.36
ABCB1 P08183 1/20 0.35
KEAP1 Q14145 1/20 0.35
NFE2L2 Q16236 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC2 Q92769 1/20 0.35
P2RX7 Q99572 1/20 0.35
ECE1 P42892 1/20 0.35
TLR2 O60603 1/20 0.34
TLR1 Q15399 1/20 0.34
HTT P42858 1/20 0.34
PKM P14618 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9519252 0.93 ATM (0.38) DPP8DPP9ATMTDP1ALDH1A1
SCHEMBL9521116 0.89 ATM (0.40) ATMTDP1ALDH1A1NPC1RAB9A
SCHEMBL9519248 0.87 ATM (0.41) ATMTDP1NPC1RAB9AECE1
SCHEMBL9519184 0.85 CTSL (0.36) DPP8DPP9ATMTDP1ALDH1A1
SCHEMBL8758724 0.85 ATM (0.44) ATMTDP1ALDH1A1NPC1RAB9A
SCHEMBL8759542 0.85 ATM (0.44) ATMTDP1ALDH1A1NPC1RAB9A
SCHEMBL9519178 0.84 DPP8 (0.46) DPP8DPP9ATMTDP1ALDH1A1
SCHEMBL9520708 0.84 DPP8 (0.46) DPP8DPP9ATMTDP1ALDH1A1
SCHEMBL9519787 0.84 ATM (0.41) ATMTDP1ALDH1A1NPC1RAB9A
SCHEMBL9519209 0.82 HTT (0.40) ATMTDP1ALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0280771-B1 3-Pyrrolidinylthio-1-azabicyclo[3.2.0]hept-2-ene-2-carboxylic acid derivatives and processes for the preparation thereof FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1993-07-28 EP disclosed
US-5061804-A 3-thiopyrrolidine as chemical intermediates FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1991-10-29 US disclosed