SCHEMBL9521928

SCHEMBL9521928

COc1c(N)ccc(F)c1N1CCN(C)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MAPT P10636 3/20 0.41
KDM4E B2RXH2 2/20 0.41
GAA P10253 2/20 0.41
PTK2B Q14289 2/20 0.41
MAPK1 P28482 1/20 0.41
HTT P42858 1/20 0.41
RECQL P46063 1/20 0.41
ADRA2C P18825 3/20 0.40
POLB P06746 1/20 0.40
GFER P55789 1/20 0.39
KMT2A Q03164 1/20 0.39
ESR2 Q92731 1/20 0.39
DRD2 P14416 2/20 0.38
DRD3 P35462 2/20 0.38
MAP4K1 Q92918 1/20 0.37
HRH4 Q9H3N8 1/20 0.36
SLC6A3 Q01959 1/20 0.36
RPS6KA3 P51812 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27565044 0.83 DRD2 (0.46) ALDH1A1MAPTKDM4EGAAPTK2B
SCHEMBL25530113 0.81 MAP4K4 (0.37) SLC6A3HTR1A
SCHEMBL12714783 0.78 ALDH1A1 (0.54) ALDH1A1L3MBTL1MAPTKDM4EGAA
SCHEMBL9525829 0.75 MAPT (0.41) ALDH1A1L3MBTL1MAPTKDM4EGAA
SCHEMBL25529972 0.75
SCHEMBL24620323 0.74 ALDH1A1 (0.49) ALDH1A1L3MBTL1MAPTKDM4EGAA
SCHEMBL30833057 0.74 ALDH1A1 (0.49) ALDH1A1L3MBTL1MAPTKDM4EGAA
SCHEMBL24054860 0.73 ADRA2C (0.53) ALDH1A1L3MBTL1MAPTKDM4EGAA
SCHEMBL9523246 0.71 DRD3 (0.56) ALDH1A1KDM4EMAPK1KMT2ADRD2
SCHEMBL3433100 0.71 ADRA2C (0.64) ALDH1A1L3MBTL1MAPTKDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0249043-B1 QUINOLINECARBOXYLIC ACID DERIVATIVES NIPPON SHINYAKU COMPANY, LIMITED (JP) 1993-08-04 EP disclosed
US-5086049-A Bactericides NIPPONSHINYAKU CO., LTD. (JP) 1992-02-04 US disclosed
US-4843070-A BACTERIDCIDES, FUNGICIDES NIPPON SHINYAKU CO., LTD. (JP) 1989-06-27 US disclosed
EP-0249043-A2 Quinolinecarboxylic acid derivatives NIPPON SHINYAKU COMPANY, LIMITED (JP) 1987-12-16 EP disclosed