SCHEMBL9522767

SCHEMBL9522767

COc1cnc2sc(S(=O)(=O)Cc3ccccc3)nn2c1=O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.42
MEN1 O00255 1/20 0.42
RXFP1 Q9HBX9 1/20 0.42
RAB9A P51151 2/20 0.39
NPC1 O15118 2/20 0.39
MITF O75030 1/20 0.39
PAX8 Q06710 1/20 0.39
ALDH1A1 P00352 4/20 0.39
MAPT P10636 4/20 0.39
NPSR1 Q6W5P4 1/20 0.39
MTOR P42345 1/20 0.39
P2RX7 Q99572 2/20 0.39
KDM4E B2RXH2 2/20 0.38
APLNR P35414 1/20 0.38
RECQL P46063 1/20 0.38
BLM P54132 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
SAE1 Q9UBE0 1/20 0.38
UBA2 Q9UBT2 1/20 0.38
NR1I2 O75469 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9521967 0.85 MAPT (0.41) KMT2AMEN1RXFP1RAB9ANPC1
SCHEMBL9522162 0.83 RAB9A (0.43) KMT2AMEN1RAB9ANPC1MITF
SCHEMBL9523127 0.83 ALDH1A1 (0.38) KMT2AMEN1RXFP1RAB9ANPC1
SCHEMBL9776505 0.81 ALDH1A1 (0.40) KMT2AMEN1RXFP1RAB9AALDH1A1
SCHEMBL10372931 0.80 KDM4E (0.50) KMT2AMEN1RAB9ANPC1ALDH1A1
SCHEMBL9521955 0.79 LOX (0.38) KMT2AMEN1RXFP1RAB9ANPC1
SCHEMBL9776524 0.77 TXNRD1 (0.44) KMT2AMEN1RXFP1RAB9AALDH1A1
SCHEMBL9532673 0.76 SOAT1 (0.44) KMT2AMEN1ALDH1A1MAPTHPGD
SCHEMBL9533205 0.76 SOAT1 (0.44) KMT2AMEN1ALDH1A1MAPTHPGD
SCHEMBL9523984 0.76 PKM (0.62) RAB9ANPC1ALDH1A1MAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0242690-B1 5H-1,3,4-Thiadiazolo[3,2-a]pyrimidin-5-one derivatives and agricultural-horticultural fungicide composition containing the same KUMIAI CHEMICAL INDUSTRY CO., LTD. (JP) 1993-06-30 EP claimed
EP-0242690-A2 5H-1,3,4-Thiadiazolo[3,2-a]pyrimidin-5-one derivatives and agricultural-horticultural fungicide composition containing the same KUMIAI CHEMICAL INDUSTRY CO., LTD. (JP) 1987-10-28 EP claimed
JP-63045286-A None JP disclosed
EP-0242690-B1 5H-1,3,4-Thiadiazolo[3,2-a]pyrimidin-5-one derivatives and agricultural-horticultural fungicide composition containing the same KUMIAI CHEMICAL INDUSTRY CO., LTD. (JP) 1993-06-30 EP disclosed
US-4985432-A 5H-1,3,4-thiadiazolo(3,2-A)pyrimidin-5-one derivatives and agricultural-horticultural fungicide composition containing the same KUMIAI CHEMICAL INDUSTRY CO., LTD. (JP) 1991-01-15 US disclosed
JP-S6345286-A 5H-1,3,4-THIADIAZOLO(3,2-A)PYRIMIDIN-5-ONE DERIVATIVE AND AGRICULTURAL AND HORTZCULTURAL GERMICIDE CONTAINING SAID COMPOUND AS ACTIVE INGREDIENT KUMIAI CHEM IND CO LTD 1988-02-26 JP disclosed
EP-0242690-A2 5H-1,3,4-Thiadiazolo[3,2-a]pyrimidin-5-one derivatives and agricultural-horticultural fungicide composition containing the same KUMIAI CHEMICAL INDUSTRY CO., LTD. (JP) 1987-10-28 EP disclosed