SCHEMBL9524637

SCHEMBL9524637

CC1(C)C=C(c2ccc(Cl)cn2)c2cc(C#N)ccc2O1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 3/20 0.39
ABCC9 O60706 11/20 0.36
BACE1 P56817 1/20 0.34
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
ABCC8 Q09428 1/20 0.33
KCNJ11 Q14654 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9524497 0.87 GRM5 (0.39) GRM5ABCC9PDE4APDE4BPDE4C
SCHEMBL9528002 0.86 KDM1A (0.36) GRM5ABCC9PDE4APDE4BPDE4C
SCHEMBL9525564 0.86 KDM1A (0.36) GRM5ABCC9BACE1PDE4APDE4B
SCHEMBL9628243 0.86 PDE4A (0.34) GRM5ABCC9BACE1PDE4APDE4B
SCHEMBL9527814 0.83 PDE4A (0.34) ABCC9PDE4APDE4BPDE4CPDE4D
SCHEMBL9527764 0.83 RARA (0.40) GRM5ABCC9BACE1PDE4APDE4B
SCHEMBL9525005 0.83 GABRA1 (0.38) ABCC9BACE1PDE4APDE4BPDE4C
SCHEMBL9523558 0.82 RARA (0.42) ABCC9PDE4APDE4BPDE4CPDE4D
Hydrochloric Acid SCHEMBL9627192 0.82 PDE4A (0.34) ABCC9PDE4APDE4BPDE4CPDE4D
SCHEMBL9527648 0.82 ABCC9 (0.39) ABCC9PDE4APDE4BPDE4CPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0298452-B1 2H-1-BENZOPYRANE DERIVATIVES SUBSTITUTED IN POSITION 4 BY ARYL OR N-HETEROARYL F. HOFFMANN-LA ROCHE AG (CH) 1993-06-30 EP disclosed
US-5118694-A Hypotensive agents; treatment for cardiovascular and muscular disorders HOFFMANN-LA ROCHE INC. (US) 1992-06-02 US disclosed
US-4971982-A HYPOTENSIVE AGENTS, CARDIOVASCULAR DISORDERS, SMOOTH MUSCLE DISORDERS HOFFMANN-LA ROCHE INC. (US) 1990-11-20 US disclosed
EP-0298452-A2 2H-1-benzopyrane derivatives substituted in position 4 by aryl or N-heteroaryl F. HOFFMANN-LA ROCHE AG (CH) 1989-01-11 EP disclosed