SCHEMBL9628243

SCHEMBL9628243

CC1(C)C=C(c2ccc(I)cn2)c2cc(C#N)ccc2O1

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34
KDM1A O60341 2/20 0.32
MAOA P21397 1/20 0.32
ABCC9 O60706 1/20 0.31
ABCB1 P08183 1/20 0.31
GRM5 P41594 1/20 0.31
BACE1 P56817 1/20 0.30
MALT1 Q9UDY8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9524497 0.87 GRM5 (0.39) PDE4APDE4BPDE4CPDE4DKDM1A
SCHEMBL9528002 0.86 KDM1A (0.36) PDE4APDE4BPDE4CPDE4DKDM1A
SCHEMBL9525564 0.86 KDM1A (0.36) PDE4APDE4BPDE4CPDE4DKDM1A
SCHEMBL9524637 0.86 GRM5 (0.39) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL9527764 0.83 RARA (0.40) PDE4APDE4BPDE4CPDE4DKDM1A
SCHEMBL9527814 0.83 PDE4A (0.34) PDE4APDE4BPDE4CPDE4DKDM1A
SCHEMBL9525005 0.83 GABRA1 (0.38) PDE4APDE4BPDE4CPDE4DABCC9
SCHEMBL9523558 0.82 RARA (0.42) PDE4APDE4BPDE4CPDE4DABCC9
Hydrochloric Acid SCHEMBL9627192 0.82 PDE4A (0.34) PDE4APDE4BPDE4CPDE4DKDM1A
SCHEMBL9527648 0.82 ABCC9 (0.39) PDE4APDE4BPDE4CPDE4DABCC9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5118694-A Hypotensive agents; treatment for cardiovascular and muscular disorders HOFFMANN-LA ROCHE INC. (US) 1992-06-02 US disclosed
US-4971982-A HYPOTENSIVE AGENTS, CARDIOVASCULAR DISORDERS, SMOOTH MUSCLE DISORDERS HOFFMANN-LA ROCHE INC. (US) 1990-11-20 US disclosed