SCHEMBL9524639

SCHEMBL9524639

COC(=O)c1cc2c(cc(C=O)c3ccccc32)s1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 6/20 0.49
ALDH1A1 P00352 6/20 0.49
MCL1 Q07820 1/20 0.44
KDM4E B2RXH2 5/20 0.41
HSD17B10 Q99714 3/20 0.41
POLB P06746 1/20 0.41
MAPK1 P28482 3/20 0.41
LMNA P02545 2/20 0.41
RPS6KB1 P23443 1/20 0.41
CSNK1D P48730 1/20 0.41
GSK3A P49840 1/20 0.41
GSK3B P49841 1/20 0.41
DYRK1A Q13627 1/20 0.41
NTRK2 Q16620 1/20 0.41
AURKB Q96GD4 1/20 0.41
CSNK2A2 P19784 2/20 0.41
CSNK2B P67870 2/20 0.41
CSNK2A1 P68400 2/20 0.41
PAK4 O96013 1/20 0.41
AKT1 P31749 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9526677 0.85 BCL2L1 (0.47) HPGDALDH1A1MCL1KDM4EMAPK1
SCHEMBL9431255 0.80 HDAC3 (0.49) HPGDALDH1A1KDM4EHSD17B10POLB
SCHEMBL9526183 0.80 HPGD (0.55) HPGDALDH1A1MCL1KDM4EHSD17B10
SCHEMBL9431295 0.75 ALDH1A1 (0.60) HPGDALDH1A1KDM4EHSD17B10POLB
SCHEMBL9978633 0.72 MCL1 (0.59) HPGDALDH1A1MCL1KDM4EHSD17B10
SCHEMBL30881132 0.71 ALOX15 (0.48) HPGDALDH1A1KDM4EHSD17B10POLB
SCHEMBL8329863 0.71 HDAC3 (0.51) HPGDALDH1A1KDM4EHSD17B10POLB
SCHEMBL828305 0.70 SLC9A1 (0.60) HPGDALDH1A1KDM4EHSD17B10POLB
SCHEMBL10080788 0.70 HCRTR1 (0.49) ALDH1A1MCL1LMNAALOX15TSHR
SCHEMBL27297693 0.70 ERN1 (0.46) HPGDALDH1A1KDM4EHSD17B10POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0183439-B1 POLYCYCLIC COMPOUNDS, THEIR PREPARATION AND USE AND FORMULATIONS CONTAINING THEM THE WELLCOME FOUNDATION LIMITED (GB) 1993-02-03 EP disclosed
US-5075455-A Microbiocides, antitumor agents BURROUGHS WELLCOME CO. (US) 1991-12-24 US disclosed
US-5049581-A Dibenzofurans having anti-tumor activity BURROUGHS WELLCOME CO. (US) 1991-09-17 US disclosed
US-5017600-A Antitumor BURROUGHS WELLCOME CO. (US) 1991-05-21 US disclosed
US-5008286-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1991-04-16 US disclosed
US-4970227-A ANTITUMOR BURROUGHS WELLCOME CO. (US) 1990-11-13 US disclosed
US-4965285-A ANTITUMOR AGENTS BURROUGHS WELLCOME CO. (US) 1990-10-23 US disclosed
US-4866070-A ANTITUMOR AGENT BURROUGHS WELLCOME CO. (US) 1989-09-12 US disclosed
EP-0183439-A2 Polycyclic compounds, their preparation and use and formulations containing them THE WELLCOME FOUNDATION LIMITED (GB) 1986-06-04 EP disclosed