SCHEMBL9524734

SCHEMBL9524734

CN(C)CC1COC2(CCN(NC(=O)OCc3ccccc3)CC2)O1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 6/20 0.41
CHRM4 P08173 6/20 0.41
CHRM5 P08912 6/20 0.41
CHRM1 P11229 6/20 0.41
CHRM3 P20309 6/20 0.41
LIPE Q05469 1/20 0.39
TMEM97 Q5BJF2 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
HTR1A P08908 5/20 0.38
ADRA1D P25100 5/20 0.38
ADRA1A P35348 5/20 0.38
ADRA1B P35368 5/20 0.38
CCR1 P32246 2/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9524247 0.88 HTR1A (0.38) LIPETMEM97SIGMAR1HTR1AADRA1D
SCHEMBL9523669 0.87 LIPE (0.40) LIPETMEM97SIGMAR1HTR1AADRA1D
SCHEMBL9384884 0.81 LIPE (0.40) LIPETMEM97SIGMAR1HTR1ACCR1
SCHEMBL25819360 0.79 LIPE (0.50) LIPEALDH1A1
SCHEMBL9527774 0.77 SYK (0.41) LIPESIGMAR1HTR1AADRA1DADRA1A
Benzyl Carbamate SCHEMBL9527492 0.74 CHRM2 (0.39) CHRM2CHRM4CHRM5CHRM1CHRM3
SCHEMBL4416797 0.71 MEN1 (0.51) CHRM4TMEM97SIGMAR1HTR1AADRA1D
SCHEMBL3673656 0.70 ALDH1A1 (0.49) LIPEALDH1A1
SCHEMBL5141506 0.70 KDM4E (0.43) LIPEALDH1A1
SCHEMBL30981534 0.69 LIPE (0.47) LIPEALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0562042-A1 QUINOLINE, NAPHTHYRIDINE AND PYRIDOBENZOXAZINE DERIVATIVES ABBOTT LABORATORIES (US) 1993-09-29 EP disclosed
US-5137892-A Bactericides ABBOTT LABORATORIES (US) 1992-08-11 US disclosed
WO-1992010191-A1 QUINOLINE, NAPHTHYRIDINE AND PYRIDOBENZOXAZINE DERIVATIVES ABBOTT LABORATORIES (US) 1992-06-25 WO disclosed