SCHEMBL9525174

SCHEMBL9525174

O=C(NCCOC(=O)C1NCCc2ccccc21)OCCN(C(=O)c1cncc(Br)c1)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
POLB P06746 2/20 0.38
TAS1R3 Q7RTX0 1/20 0.38
TAS1R1 Q7RTX1 1/20 0.38
TAS1R2 Q8TE23 1/20 0.38
TSHR P16473 2/20 0.35
NPSR1 Q6W5P4 1/20 0.35
ROCK2 O75116 1/20 0.34
SMN1; SMN2 Q16637 4/20 0.34
ALDH1A1 P00352 2/20 0.34
OPRM1 P35372 2/20 0.33
LMNA P02545 2/20 0.33
MAPT P10636 2/20 0.33
HTT P42858 2/20 0.33
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
KDM4C Q9H3R0 1/20 0.31
HPGD P15428 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9524781 0.91 NPC1 (0.38) NPC1RAB9APOLBTAS1R3TAS1R1
SCHEMBL9525693 0.88 POLB (0.35) NPC1RAB9APOLBTAS1R3TAS1R1
SCHEMBL9526317 0.87 POLB (0.35) NPC1RAB9APOLBTAS1R3TAS1R1
SCHEMBL9528461 0.87 NPC1 (0.37) NPC1RAB9APOLBTAS1R3TAS1R1
Hydrochloric Acid SCHEMBL9525305 0.84 TSHR (0.33) TSHRNPSR1ROCK2OPRM1SLC18A2
SCHEMBL9524060 0.82 OPRM1 (0.37) TSHRNPSR1ROCK2SMN1; SMN2OPRM1
SCHEMBL9525136 0.82 OPRM1 (0.37) RAB9ATSHRNPSR1ROCK2SMN1; SMN2
SCHEMBL9525702 0.81 TSHR (0.42) POLBTAS1R3TAS1R1TAS1R2TSHR
SCHEMBL9528525 0.80 POLB (0.34) POLBTAS1R3TAS1R1TAS1R2TSHR
SCHEMBL9526039 0.80 NPC1 (0.42) NPC1RAB9APOLBTAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301751-B1 PYRIDINIUM DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-03-10 EP disclosed
US-4962113-A PLATELET ACTIVATING FACTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1990-10-09 US disclosed
EP-0301751-A1 Pyridinium derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-02-01 EP disclosed