SCHEMBL9526317

SCHEMBL9526317

O=C(NCC(OC(=O)C1NCCc2ccccc21)c1ccccc1)OCCN(C(=O)c1cncc(Br)c1)c1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.35
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
TAS1R2 Q8TE23 1/20 0.35
TSHR P16473 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
ROCK2 O75116 1/20 0.32
MAPT P10636 2/20 0.32
LMNA P02545 1/20 0.32
HTT P42858 1/20 0.32
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
OPRM1 P35372 1/20 0.31
SMN1; SMN2 Q16637 2/20 0.30
ALDH1A1 P00352 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9525693 0.91 POLB (0.35) POLBTAS1R3TAS1R1TAS1R2TSHR
SCHEMBL9525174 0.87 NPC1 (0.38) POLBTAS1R3TAS1R1TAS1R2TSHR
Hydrochloric Acid SCHEMBL9528195 0.86 TSHR (0.30) TSHRNPSR1
SCHEMBL9525947 0.81 NPC1 (0.39) POLBTSHRNPSR1MAPTLMNA
SCHEMBL9524781 0.80 NPC1 (0.38) POLBTAS1R3TAS1R1TAS1R2TSHR
SCHEMBL9528461 0.79 NPC1 (0.37) POLBTAS1R3TAS1R1TAS1R2TSHR
SCHEMBL9526212 0.78 SMN1; SMN2 (0.39) POLBMAPTLMNAHTTNPC1
SCHEMBL9528525 0.78 POLB (0.34) POLBTAS1R3TAS1R1TAS1R2TSHR
Hydrochloric Acid SCHEMBL9525127 0.77 TSHR (0.31) TSHRNPSR1OPRM1
SCHEMBL9525702 0.77 TSHR (0.42) POLBTAS1R3TAS1R1TAS1R2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301751-B1 PYRIDINIUM DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-03-10 EP disclosed
US-4962113-A PLATELET ACTIVATING FACTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1990-10-09 US disclosed
EP-0301751-A1 Pyridinium derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-02-01 EP disclosed