SCHEMBL9528461

SCHEMBL9528461

O=C(CCN(C(=O)c1cncc(Br)c1)c1ccccc1)NCCCOC(=O)C1NCCc2ccccc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
POLB P06746 2/20 0.37
TAS1R3 Q7RTX0 1/20 0.37
TAS1R1 Q7RTX1 1/20 0.37
TAS1R2 Q8TE23 1/20 0.37
TSHR P16473 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
ROCK2 O75116 1/20 0.34
SMN1; SMN2 Q16637 4/20 0.33
ALDH1A1 P00352 3/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C19 P33261 1/20 0.33
OPRM1 P35372 1/20 0.33
LMNA P02545 2/20 0.32
MAPT P10636 2/20 0.32
SLC6A2 P23975 1/20 0.32
SLC6A4 P31645 1/20 0.32
HTT P42858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9524781 0.96 NPC1 (0.38) NPC1RAB9APOLBTAS1R3TAS1R1
SCHEMBL9525136 0.87 OPRM1 (0.37) RAB9ATSHRNPSR1ROCK2SMN1; SMN2
SCHEMBL9524060 0.87 OPRM1 (0.37) TSHRNPSR1ROCK2SMN1; SMN2OPRM1
SCHEMBL9525174 0.87 NPC1 (0.38) NPC1RAB9APOLBTAS1R3TAS1R1
SCHEMBL9528525 0.85 POLB (0.34) POLBTAS1R3TAS1R1TAS1R2TSHR
SCHEMBL9525702 0.83 TSHR (0.42) POLBTAS1R3TAS1R1TAS1R2TSHR
SCHEMBL9528889 0.81 TSHR (0.33) TSHRNPSR1ROCK2OPRM1SLC6A2
Hydrochloric Acid SCHEMBL9523922 0.80 TSHR (0.33) TSHRNPSR1ROCK2OPRM1SLC6A2
SCHEMBL9525693 0.80 POLB (0.35) NPC1RAB9APOLBTAS1R3TAS1R1
SCHEMBL9526317 0.79 POLB (0.35) NPC1RAB9APOLBTAS1R3TAS1R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301751-B1 PYRIDINIUM DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-03-10 EP disclosed
EP-0301751-A1 Pyridinium derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-02-01 EP disclosed