SCHEMBL9525362

SCHEMBL9525362

O=C(CCN(C(=O)c1cncc(Br)c1)c1ccccc1)Nc1cccc2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BLM P54132 1/20 0.43
ALDH1A1 P00352 2/20 0.43
CYP1A2 P05177 2/20 0.42
CYP2C19 P33261 2/20 0.42
HDAC4 P56524 2/20 0.42
KDR P35968 2/20 0.42
HDAC3 O15379 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC7 Q8WUI4 1/20 0.42
HDAC2 Q92769 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC11 Q96DB2 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HDAC9 Q9UKV0 1/20 0.42
HDAC5 Q9UQL6 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HTT P42858 2/20 0.41
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9528510 0.95 SMN1; SMN2 (0.40) BLMALDH1A1CYP1A2CYP2C19HDAC4
SCHEMBL9525706 0.92 CYP1A2 (0.41) BLMALDH1A1CYP1A2CYP2C19HDAC4
SCHEMBL9524974 0.87 ALDH1A1 (0.41) BLMALDH1A1KDRSMN1; SMN2MEN1
SCHEMBL9525433 0.86 EPHX1 (0.45) ALDH1A1CYP1A2CYP2C19KDRSMN1; SMN2
SCHEMBL9524184 0.86 ALDH1A1 (0.47) BLMALDH1A1CYP1A2CYP2C19KDR
SCHEMBL9525296 0.83 ALDH1A1 (0.43) BLMALDH1A1KDRSMN1; SMN2MEN1
SCHEMBL9526036 0.83 ALDH1A1 (0.43) BLMALDH1A1KDRSMN1; SMN2MEN1
SCHEMBL9525975 0.82 SMN1; SMN2 (0.43) ALDH1A1HDAC4KDRHDAC3HDAC1
SCHEMBL9525236 0.82 ALDH1A1 (0.40) BLMALDH1A1HDAC4KDRHDAC3
SCHEMBL9525424 0.82 ALDH1A1 (0.43) BLMALDH1A1KDRSMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301751-B1 PYRIDINIUM DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-03-10 EP disclosed
US-4962113-A PLATELET ACTIVATING FACTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1990-10-09 US disclosed
EP-0301751-A1 Pyridinium derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-02-01 EP disclosed