SCHEMBL9528510

SCHEMBL9528510

O=C(CCN(C(=O)c1cncc(Br)c1)c1ccccc1)NCCC(=O)Nc1cccc2ccccc12

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.40
BLM P54132 1/20 0.39
EPHX1 P07099 1/20 0.39
ALDH1A1 P00352 2/20 0.39
HDAC4 P56524 2/20 0.39
KDR P35968 2/20 0.39
HDAC3 O15379 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C19 P33261 1/20 0.39
SIRT2 Q8IXJ6 1/20 0.38
SIRT1 Q96EB6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9525362 0.95 BLM (0.43) SMN1; SMN2BLMALDH1A1HDAC4KDR
SCHEMBL9525706 0.94 CYP1A2 (0.41) SMN1; SMN2BLMEPHX1ALDH1A1HDAC4
SCHEMBL9525433 0.92 EPHX1 (0.45) SMN1; SMN2EPHX1ALDH1A1KDRCYP1A2
SCHEMBL9524974 0.89 ALDH1A1 (0.41) SMN1; SMN2BLMALDH1A1KDRSIRT2
SCHEMBL9525975 0.85 SMN1; SMN2 (0.43) SMN1; SMN2ALDH1A1HDAC4KDRHDAC3
SCHEMBL9525236 0.84 ALDH1A1 (0.40) SMN1; SMN2BLMALDH1A1HDAC4KDR
SCHEMBL9524780 0.83 FLT3 (0.43) SMN1; SMN2ALDH1A1KDRCYP1A2CYP2C19
SCHEMBL9525116 0.82 SMN1; SMN2 (0.46) SMN1; SMN2ALDH1A1HDAC1HDAC6HTT
Hydrochloric Acid SCHEMBL9525275 0.82 EPHX1 (0.40) EPHX1ALDH1A1HDAC4HDAC3HDAC1
SCHEMBL9524016 0.81 ALDH1A1 (0.41) SMN1; SMN2BLMEPHX1ALDH1A1KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301751-B1 PYRIDINIUM DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-03-10 EP disclosed
US-4962113-A PLATELET ACTIVATING FACTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1990-10-09 US disclosed
EP-0301751-A1 Pyridinium derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-02-01 EP disclosed