SCHEMBL9525975

SCHEMBL9525975

O=C(CCN(C(=O)c1cncc(Br)c1)c1ccccc1)NCCNC(=O)c1cccc2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.43
POLB P06746 1/20 0.42
ALDH1A1 P00352 5/20 0.42
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
GLA P06280 1/20 0.40
PPARG P37231 1/20 0.39
HPGD P15428 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
HDAC1 Q13547 2/20 0.38
HDAC6 Q9UBN7 2/20 0.38
HDAC2 Q92769 2/20 0.38
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9524780 0.85 FLT3 (0.43) SMN1; SMN2POLBALDH1A1NPC1RAB9A
SCHEMBL9528510 0.85 SMN1; SMN2 (0.40) SMN1; SMN2POLBALDH1A1NPC1RAB9A
SCHEMBL9525116 0.83 SMN1; SMN2 (0.46) SMN1; SMN2POLBALDH1A1NPC1RAB9A
SCHEMBL9525362 0.82 BLM (0.43) SMN1; SMN2ALDH1A1NPC1RAB9AMEN1
SCHEMBL9525706 0.82 CYP1A2 (0.41) SMN1; SMN2POLBALDH1A1NPC1RAB9A
SCHEMBL9524974 0.81 ALDH1A1 (0.41) SMN1; SMN2POLBALDH1A1NPC1RAB9A
Hydrochloric Acid SCHEMBL9524291 0.81 HDAC1 (0.37) ALDH1A1PPARGHPGDMEN1KMT2A
SCHEMBL9527984 0.81 SMN1; SMN2 (0.46) SMN1; SMN2POLBALDH1A1NPC1RAB9A
SCHEMBL9525433 0.81 EPHX1 (0.45) SMN1; SMN2POLBALDH1A1NPC1MEN1
SCHEMBL9525795 0.79 SMN1; SMN2 (0.46) SMN1; SMN2POLBALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301751-B1 PYRIDINIUM DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-03-10 EP disclosed
US-4962113-A PLATELET ACTIVATING FACTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1990-10-09 US disclosed
EP-0301751-A1 Pyridinium derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-02-01 EP disclosed