SCHEMBL9526164

SCHEMBL9526164

Sc1nc(-c2cnc3ccccc3c2)n[nH]1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 3/20 0.49
PDGFRA P16234 3/20 0.49
CYP2A6 P11509 1/20 0.46
NISCH Q9Y2I1 1/20 0.46
BIRC5 O15392 1/20 0.45
PIK3CD O00329 1/20 0.44
PIK3CA P42336 1/20 0.44
MAP4K4 O95819 1/20 0.43
CSNK1G2 P78368 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
MKNK2 Q9HBH9 1/20 0.43
MAP4K5 Q9Y4K4 1/20 0.43
TOP2A P11388 1/20 0.43
TOP2B Q02880 1/20 0.43
HPGDS O60760 1/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
CYP1A2 P05177 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL657644 0.77 NR1H2 (0.61) HPGDSCYP1A2NPC1MAPTRAB9A
SCHEMBL32667946 0.75 PDGFRB (0.77) PDGFRBPDGFRACYP2A6NISCHBIRC5
SCHEMBL2772360 0.75 PDGFRB (0.77) PDGFRBPDGFRACYP2A6NISCHBIRC5
SCHEMBL24412080 0.74 PDGFRB (0.65) PDGFRBPDGFRACYP2A6NISCHBIRC5
SCHEMBL4170881 0.73 HPGDS (0.61) PDGFRBPDGFRACYP2A6NISCHBIRC5
SCHEMBL17944740 0.71 PDGFRB (0.61) PDGFRBPDGFRACYP2A6NISCHBIRC5
SCHEMBL29179966 0.71 CYP1A2 (0.63) PDGFRBPDGFRACYP2A6NISCHBIRC5
SCHEMBL10051400 0.70 PDGFRB (0.54) PDGFRBPDGFRACYP2A6NISCHBIRC5
SCHEMBL6985344 0.70 POLB (0.57) PDGFRBPDGFRACYP2A6NISCHBIRC5
SCHEMBL25439863 0.70 CYP1A2 (0.56) PDGFRBPDGFRACYP2A6NISCHBIRC5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276793-B1 3-ARYL-5-ALKYLTHIO-4H-1,2,4-TRIAZOLES MERRELL DOW PHARMACEUTICALS INC. (US) 1993-06-16 EP disclosed
EP-0226755-B1 5-HETEROCYCLIC-3H-1,2,4-TRIAZOLE-3-THIONES AND THEIR USE AS ANTIDEPRESSANTS MERRELL DOW PHARMACEUTICALS INC. (US) 1991-08-14 EP disclosed