SCHEMBL949313

SCHEMBL949313

Nc1cc(-c2nnn[nH]2)ccc1Cc1ccc2ccccc2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MPO P05164 1/20 0.42
ALOX5 P09917 1/20 0.40
CTRC Q99895 1/20 0.37
CHEK2 O96017 1/20 0.36
CYP2D6 P10635 1/20 0.36
NFKB1 P19838 1/20 0.36
TAAR1 Q96RJ0 1/20 0.36
BACE1 P56817 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
PDE10A Q9Y233 2/20 0.34
IKBKB O14920 1/20 0.33
TBXA2R P21731 1/20 0.33
PTGER4 P35408 1/20 0.33
PTGFR P43088 1/20 0.33
PTGER3 P43115 1/20 0.33
PTGER2 P43116 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL670906 0.78 NOTUM (0.42) ALOX5ADORA2AADORA1IKBKB
SCHEMBL952623 0.76 MPO (0.37) MPOALOX5CHEK2CYP2D6NFKB1
SCHEMBL6775919 0.74 DHFR (0.42) ALOX5NFKB1ADORA2AADORA1IKBKB
SCHEMBL1247974 0.72 CYP2D6 (0.46) MPOALOX5CYP2D6NFKB1TAAR1
SCHEMBL949314 0.71 INSR (0.44) ADORA2AADORA1
SCHEMBL949966 0.71 MC5R (0.36) HDAC1
SCHEMBL22666679 0.70 ALOX5 (0.53) MPOALOX5CTRCCYP2D6NFKB1
SCHEMBL21371042 0.70 ALOX5 (0.50) MPOALOX5CTRCCYP2D6NFKB1
Hydrochloric Acid SCHEMBL16176998 0.69 TDP1 (0.46) NFKB1
SCHEMBL6955273 0.68 CALM1 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011006935-A2 TETRAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2011-01-20 WO disclosed