SCHEMBL9526686

SCHEMBL9526686

CCCC(c1ccc(C(=O)O)cc1OC)c1c[nH]c2ccc(CC3CCN(C)C3=O)cc12

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.36
RAB9A P51151 1/20 0.36
SLC6A4 P31645 1/20 0.34
ROCK2 O75116 1/20 0.34
FFAR1 O14842 1/20 0.33
GPR84 Q9NQS5 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRB2 P47870 1/20 0.33
TSHR P16473 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HTT P42858 1/20 0.33
TAAR1 Q96RJ0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9527469 0.95 NPC1 (0.35) NPC1RAB9ASLC6A4ROCK2GABRA1
SCHEMBL9527468 0.94 B3GAT3 (0.35) RAB9A
SCHEMBL9527712 0.92 NPC1 (0.35) NPC1RAB9AROCK2FFAR1GPR84
SCHEMBL9526771 0.92 NPC1 (0.34) NPC1RAB9ASLC6A4ROCK2FFAR1
SCHEMBL9526764 0.90 NPC1 (0.37) NPC1RAB9AROCK2SMN1; SMN2TSHR
SCHEMBL9527749 0.89 HTR1D (0.35) RAB9ASLC6A4GABRA1GABRB2ALDH1A1
SCHEMBL9528145 0.88 KDM2B (0.35) NPC1RAB9ASLC6A4FFAR1GPR84
SCHEMBL9527280 0.86 B3GAT3 (0.34) RAB9A
SCHEMBL9527214 0.85 HTR7 (0.34) RAB9AROCK2GPR84SMN1; SMN2ALDH1A1
SCHEMBL9527270 0.85 MEN1 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0337767-B1 CYCLIC AMIDES ICI AMERICAS INC. (US) 1993-01-13 EP disclosed
US-5047402-A Leukotriene Antagonists ICI AMERICAS INC. (US) 1991-09-10 US disclosed
EP-0337767-A1 Cyclic amides ICI AMERICAS INC. (US) 1989-10-18 EP disclosed