SCHEMBL9526764

SCHEMBL9526764

COc1cc(C(=O)O)ccc1C(C)c1c[nH]c2ccc(CC3CCN(C)C3=O)cc12

nearest known ligand 0.38

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.37
RAB9A P51151 1/20 0.37
ROCK2 O75116 1/20 0.35
MTNR1A P48039 1/20 0.34
MTNR1B P49286 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
TRPV1 Q8NER1 1/20 0.33
KDM4E B2RXH2 1/20 0.33
TSHR P16473 1/20 0.33
LMNA P02545 1/20 0.33
GAA P10253 1/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9526859 0.93 B3GAT3 (0.36) RAB9AROCK2MTNR1AMTNR1BTRPV1
SCHEMBL9526830 0.91 NPC1 (0.35) NPC1RAB9AROCK2MTNR1AMTNR1B
SCHEMBL9526686 0.90 NPC1 (0.36) NPC1RAB9AROCK2SMN1; SMN2TSHR
SCHEMBL9527469 0.85 NPC1 (0.35) NPC1RAB9AROCK2MTNR1AMTNR1B
SCHEMBL9528261 0.85 PTPN5 (0.35) ROCK2KDM4E
SCHEMBL9527977 0.84 CYSLTR1 (0.41)
SCHEMBL9527665 0.83 B3GAT3 (0.35) RAB9AROCK2MTNR1AMTNR1BTRPV1
SCHEMBL9527468 0.83 B3GAT3 (0.35) RAB9A
SCHEMBL9528078 0.83 CYSLTR2 (0.41) GAA
SCHEMBL9527712 0.82 NPC1 (0.35) NPC1RAB9AROCK2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0337767-B1 CYCLIC AMIDES ICI AMERICAS INC. (US) 1993-01-13 EP disclosed
US-5047402-A Leukotriene Antagonists ICI AMERICAS INC. (US) 1991-09-10 US disclosed
EP-0337767-A1 Cyclic amides ICI AMERICAS INC. (US) 1989-10-18 EP disclosed