SCHEMBL9526771

SCHEMBL9526771

CCCC(c1ccc(C(=O)O)cc1OC)c1c[nH]c2ccc(CC3CCN(CC)C3=O)cc12

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
ROCK2 O75116 1/20 0.33
FFAR1 O14842 1/20 0.33
GPR84 Q9NQS5 1/20 0.33
TSHR P16473 2/20 0.32
KDM2B Q8NHM5 1/20 0.32
SLC6A4 P31645 1/20 0.32
LMNA P02545 2/20 0.32
HTT P42858 2/20 0.32
KDM4E B2RXH2 1/20 0.32
GLA P06280 1/20 0.32
MAPT P10636 1/20 0.32
MAPK1 P28482 1/20 0.32
GAA P10253 1/20 0.31
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
HPGD P15428 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9527712 0.95 NPC1 (0.35) NPC1RAB9AROCK2FFAR1GPR84
SCHEMBL9527214 0.94 HTR7 (0.34) RAB9AROCK2GPR84KDM4EMAPK1
SCHEMBL9526686 0.92 NPC1 (0.36) NPC1RAB9AROCK2FFAR1GPR84
SCHEMBL9528145 0.89 KDM2B (0.35) NPC1RAB9AFFAR1GPR84TSHR
SCHEMBL9527280 0.89 B3GAT3 (0.34) RAB9AKDM2B
SCHEMBL9527469 0.89 NPC1 (0.35) NPC1RAB9AROCK2TSHRKDM2B
SCHEMBL9526830 0.86 NPC1 (0.35) NPC1RAB9AROCK2TSHRKDM2B
SCHEMBL9527468 0.85 B3GAT3 (0.35) RAB9A
SCHEMBL9526614 0.85 PLA2G4A (0.39) MAPTMAPK1MEN1KMT2A
SCHEMBL9528111 0.83 KDM2B (0.34) GPR84KDM2BKDM4EGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0337767-B1 CYCLIC AMIDES ICI AMERICAS INC. (US) 1993-01-13 EP disclosed
US-5047402-A Leukotriene Antagonists ICI AMERICAS INC. (US) 1991-09-10 US disclosed
EP-0337767-A1 Cyclic amides ICI AMERICAS INC. (US) 1989-10-18 EP disclosed