SCHEMBL9527735

SCHEMBL9527735

CC1(Cl)c2ccccc2CC1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.42
BLM P54132 1/20 0.42
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
SIGMAR1 Q99720 1/20 0.38
CYP3A4 P08684 2/20 0.37
MEN1 O00255 1/20 0.37
CYP2D6 P10635 1/20 0.37
ALOX15 P16050 1/20 0.37
CYP2C19 P33261 1/20 0.37
KMT2A Q03164 1/20 0.37
GRIN2D O15399 1/20 0.37
GRIN3B O60391 1/20 0.37
BCHE P06276 1/20 0.37
CHRM5 P08912 1/20 0.37
TSHR P16473 1/20 0.37
ALOX12 P18054 1/20 0.37
NFKB1 P19838 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9526996 0.76 CCR2 (0.37) LMNAMAPTCRHBPCRHR2GRIN2B
SCHEMBL1387775 0.75 GAA (0.41) LMNABLMGAAMAPTSIGMAR1
SCHEMBL6071126 0.73 GAA (0.40) LMNABLMGAAMAPTKMT2A
SCHEMBL20515884 0.73 LMNA (0.42) LMNABLMCRHBPCRHR2SIGMAR1
SCHEMBL11799039 0.72 AKR1C1 (0.40) LMNABLMGAAMAPTSIGMAR1
SCHEMBL28206833 0.71 KMT2A (0.47) LMNABLMSIGMAR1CYP3A4MEN1
SCHEMBL30715059 0.71 GAA (0.35) LMNABLMGAAMAPTCRHBP
SCHEMBL30856510 0.70 MEN1 (0.37) LMNABLMGAAMAPTSIGMAR1
SCHEMBL5835341 0.70 LMNA (0.44) LMNAMAPK1
SCHEMBL8410307 0.70 HDAC9 (0.44) GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0310745-B1 SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR PREPARATION AND USE ORION-YHTYMÄ OY (FI) 1993-01-27 EP disclosed
EP-0183492-B1 SUBSTITUTED IMIDAZOLE DERIVATIVES AND THEIR PREPARATION AND USE Farmos-Yhtyma Oy (FI) 1989-11-15 EP disclosed
EP-0310745-A2 Substituted imidazole derivatives and their preparation and use ORION-YHTYMÄ OY (FI) 1989-04-12 EP disclosed
US-4689339-A 4-dihydroinden-2-yl-, 4-tetrahydronaphth-2-yl-, and 4-dihydrobenzofuran-2-ylimidazoles, useful to block α2 -adrenergic receptors FARMOS YHTYMA OY (FI) 1987-08-25 US disclosed
EP-0183492-A1 Substituted imidazole derivatives and their preparation and use Farmos-Yhtyma Oy (FI) 1986-06-04 EP disclosed