SCHEMBL9530260

SCHEMBL9530260

COc1ccc(N2CCN(CC3CN(c4ccccc4)c4ccccc4O3)CC2)cc1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 10/20 0.53
DRD2 P14416 2/20 0.52
DRD4 P21917 1/20 0.52
ADRA2A P08913 1/20 0.51
ADRA2B P18089 1/20 0.51
ADRA2C P18825 1/20 0.51
GRM2 Q14416 1/20 0.50
ADRA1D P25100 2/20 0.48
ADRA1A P35348 2/20 0.48
ADRA1B P35368 2/20 0.48
PKM P14618 1/20 0.48
HTR1A P08908 3/20 0.47
GAA P10253 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9530044 0.89 ABCB1 (0.49) SIGMAR1DRD2DRD4ADRA2AADRA2B
Hydrochloric Acid SCHEMBL10368330 0.88 ABCB1 (0.48) SIGMAR1DRD2DRD4ADRA2AADRA2B
SCHEMBL9455118 0.85 ADRA2A (0.70) DRD2DRD4ADRA2AADRA2BADRA2C
SCHEMBL9455117 0.81 CASR (0.45) SIGMAR1DRD2DRD4ADRA2AADRA2B
SCHEMBL9455324 0.81 ADRA2A (0.66) DRD2DRD4ADRA2AADRA2BADRA2C
SCHEMBL9696810 0.80 ADRA2A (0.59) SIGMAR1ADRA2AADRA2BADRA2CADRA1D
SCHEMBL9529266 0.79 DRD2 (0.53) SIGMAR1DRD2DRD4GRM2HTR1A
SCHEMBL9455287 0.77 ADRA2A (0.59) DRD2DRD4ADRA2AADRA2BADRA2C
SCHEMBL9529716 0.76 KCNH2 (0.50) DRD2DRD4ADRA2AADRA2BADRA2C
SCHEMBL9455184 0.75 ADRA2A (0.59) DRD2DRD4ADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0359790-B1 1,4-BENZOXAZINE AND 1,4-BENZOTHIAZINE DERIVATIVES AND PROCESS FOR THEIR PREPARATION ERBA CARLO SPA (IT) 1993-11-03 EP disclosed
US-5084454-A Tranquilizers and antinausea drugs FARMITALIA CARLO ERBA S.R.L. (IT) 1992-01-28 US disclosed