SCHEMBL9532340

SCHEMBL9532340

CCc1nc(C(=O)NC2CC3CCCC(C2)N3C)c2ccccn12

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 9/20 0.59
HTR3E A5X5Y0 1/20 0.59
SLC22A2 O15244 1/20 0.59
HTR3B O95264 1/20 0.59
CHRNB2 P17787 1/20 0.59
CHRNA3 P32297 1/20 0.59
CHRNA4 P43681 1/20 0.59
KCNH2 Q12809 1/20 0.59
HTR3D Q70Z44 1/20 0.59
HTR3C Q8WXA8 1/20 0.59
SLC47A1 Q96FL8 1/20 0.59
HTR4 Q13639 5/20 0.55
CYP3A4 P08684 2/20 0.53
ALDH1A1 P00352 1/20 0.53
TSHR P16473 1/20 0.53
MAPK1 P28482 1/20 0.53
HSD17B10 Q99714 1/20 0.53
CYP2D6 P10635 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9532171 0.96 HTR4 (0.59) HTR3AHTR3ESLC22A2HTR3BCHRNB2
SCHEMBL9530584 0.78 HTR4 (0.58) HTR3AHTR3ESLC22A2HTR3BCHRNB2
Hydrochloric Acid SCHEMBL9534802 0.78 HTR4 (0.57) HTR3AHTR3ESLC22A2HTR3BCHRNB2
SCHEMBL7364679 0.75 HTR3A (0.83) HTR3AHTR3ESLC22A2HTR3BCHRNB2
SCHEMBL7497547 0.75 HTR3A (0.83) HTR3AHTR3ESLC22A2HTR3BCHRNB2
SCHEMBL9748207 0.74 HTR3A (0.53) HTR3AHTR3ESLC22A2HTR3BCHRNB2
SCHEMBL9531310 0.74 CHRNA7 (0.51) HTR3ACHRNB2CHRNA3CHRNA4HTR4
Granisetron SCHEMBL34178 0.74 HTR3A (1.00) HTR3AHTR3ESLC22A2HTR3BCHRNB2
Granisetron SCHEMBL16642163 0.74 HTR3A (1.00) HTR3AHTR3ESLC22A2HTR3BCHRNB2
Granisetron SCHEMBL445223 0.74 HTR3A (1.00) HTR3AHTR3ESLC22A2HTR3BCHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0289170-B1 AZABICYCLIC COMPOUNDS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BEECHAM GROUP PLC (GB) 1993-06-23 EP claimed
EP-0289170-A2 Azabicyclic compounds, process for their preparation and pharmaceutical compositions containing them BEECHAM GROUP PLC (GB) 1988-11-02 EP claimed
EP-0289170-B1 AZABICYCLIC COMPOUNDS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM BEECHAM GROUP PLC (GB) 1993-06-23 EP disclosed
EP-0289170-A2 Azabicyclic compounds, process for their preparation and pharmaceutical compositions containing them BEECHAM GROUP PLC (GB) 1988-11-02 EP disclosed