SCHEMBL9532459

SCHEMBL9532459

COc1ccc2[nH]cc(CCN3CCNC(CC(=O)O)C3=O)c2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.53
KDM4E B2RXH2 3/20 0.52
HTR1A P08908 5/20 0.51
RAB9A P51151 2/20 0.51
NPC1 O15118 1/20 0.51
ALDH1A1 P00352 3/20 0.50
MAPT P10636 2/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
KMT2A Q03164 3/20 0.49
MTNR1A P48039 4/20 0.48
MTNR1B P49286 3/20 0.48
CYP2D6 P10635 2/20 0.48
MEN1 O00255 2/20 0.48
CYP1A1 P04798 1/20 0.48
MPO P05164 1/20 0.48
CYP1A2 P05177 1/20 0.48
CYP3A4 P08684 1/20 0.48
HPGD P15428 1/20 0.48
NQO2 P16083 1/20 0.48
HTR2B P41595 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9528741 0.93 MTNR1A (0.48) HTR2AKDM4EHTR1ARAB9ANPC1
SCHEMBL10491444 0.89 KMT2A (0.51) HTR2AKDM4EHTR1ARAB9ANPC1
SCHEMBL9527410 0.86 SLC6A4 (0.44) HTR2AMAPTKMT2AMTNR1AMTNR1B
SCHEMBL10491382 0.82 KMT2A (0.47) HTR2AKDM4EHTR1ARAB9ANPC1
SCHEMBL9531891 0.82 HTR2A (0.43) HTR2ARAB9AMAPTKMT2AMTNR1A
SCHEMBL9529850 0.79 NPC1 (0.49) HTR2AKDM4EHTR1ARAB9ANPC1
Acetic Acid SCHEMBL9532462 0.78 HTR2A (0.56) HTR2AKDM4EHTR1ARAB9ANPC1
SCHEMBL10491419 0.78 TSHR (0.43) HTR2AHTR1ARAB9AALDH1A1MAPT
SCHEMBL30274696 0.77 HTR2A (0.57) HTR2AKDM4EHTR1ARAB9ANPC1
SCHEMBL10491380 0.75 SMN1; SMN2 (0.53) HTR2AKDM4ERAB9ANPC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0287468-B1 17-AZA-20,21-DINOREBURNAMENINE DERIVATIVES, PROCESS AND INTERMEDIATES FOR THEIR PREPARATION, THEIR USE AS MEDICAMENTS AND COMPOSITIONS CONTAINING THEM ROUSSEL-UCLAF (FR) 1993-03-10 EP disclosed
EP-0287468-A2 17-Aza-20,21-dinoreburnamenine derivatives, process and intermediates for their preparation, their use as medicaments and compositions containing them ROUSSEL-UCLAF (FR) 1988-10-19 EP disclosed