SCHEMBL9532489

SCHEMBL9532489

COc1ccc(OC)c(C(=NOCCc2ccccc2)c2cccnc2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 3/20 0.52
CYP11B2 P19099 3/20 0.52
LRRK2 Q5S007 1/20 0.45
TBXAS1 P24557 2/20 0.44
SMN1; SMN2 Q16637 3/20 0.42
TSHR P16473 2/20 0.42
KMT2A Q03164 1/20 0.42
POLB P06746 1/20 0.42
KDM4E B2RXH2 2/20 0.41
ALDH1A1 P00352 2/20 0.41
TDP1 Q9NUW8 1/20 0.41
TAAR1 Q96RJ0 1/20 0.41
ABCB1 P08183 1/20 0.41
CYP1A2 P05177 2/20 0.40
CYP3A4 P08684 2/20 0.40
MAPK1 P28482 1/20 0.40
BLM P54132 1/20 0.40
LMNA P02545 1/20 0.40
CYP2C19 P33261 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9529072 0.92 CYP11B1 (0.54) CYP11B1CYP11B2LRRK2TBXAS1SMN1; SMN2
SCHEMBL9527952 0.84 ALDH1A1 (0.49) CYP11B1CYP11B2TBXAS1KMT2APOLB
SCHEMBL9532138 0.84 TBXAS1 (0.55) CYP11B1CYP11B2TBXAS1KMT2AKDM4E
SCHEMBL9529775 0.83 TBXAS1 (0.50) CYP11B1CYP11B2TBXAS1SMN1; SMN2TSHR
SCHEMBL9532347 0.83 ABCB1 (0.53) CYP11B1CYP11B2TBXAS1SMN1; SMN2TSHR
SCHEMBL9527829 0.81 MAPK1 (0.55) TBXAS1KMT2APOLBALDH1A1CYP1A2
SCHEMBL9532300 0.81 TBXAS1 (0.57) TBXAS1SMN1; SMN2KMT2AKDM4EALDH1A1
SCHEMBL9528581 0.80 TBXAS1 (0.59) TBXAS1SMN1; SMN2KMT2AKDM4EALDH1A1
SCHEMBL9528781 0.79 MAPK1 (0.58) TBXAS1SMN1; SMN2KMT2APOLBKDM4E
SCHEMBL9531922 0.79 TBXAS1 (0.52) TBXAS1SMN1; SMN2KMT2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0366006-B1 PYRIDYLKETOXIME ETHER COMPOUND AND PHARMACEUTICAL COMPOSITION CONTAINING IT KAKEN PHARMACEUTICAL CO., LTD. (JP) 1993-09-29 EP disclosed
US-4971985-A ANTIISCHEMIC AGENTS, CARDIOVASCULAR DISORDERS KAKEN PHARMACEUTICAL CO., LTD. (JP) 1990-11-20 US disclosed