SCHEMBL9532636

SCHEMBL9532636

CCN1N=C(c2cccc3c2NC(=O)CC3)C(C)SC1=O

nearest known ligand 0.33

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 1/20 0.33
SRD5A1 P18405 1/20 0.33
CYP19A1 P11511 3/20 0.32
CYP11B1 P15538 3/20 0.32
CYP11B2 P19099 3/20 0.32
NPC1 O15118 1/20 0.31
MAPK13 O15264 1/20 0.31
MAPK12 P53778 1/20 0.31
MAPK11 Q15759 1/20 0.31
MAPK14 Q16539 1/20 0.31
DDB1 Q16531 1/20 0.31
CRBN Q96SW2 1/20 0.31
BRD4 O60885 1/20 0.30
CREBBP Q92793 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9532628 0.77 PDE3B (0.52) CYP11B1CYP11B2NPC1CRBNBRD4
SCHEMBL9527882 0.75 PDE3B (0.42) HTR2ASRD5A1CYP19A1CYP11B1CYP11B2
SCHEMBL9532290 0.71 PDE3B (0.45) CYP11B1CYP11B2NPC1
SCHEMBL29495915 0.66 GABRP (0.37) HTR2ASRD5A1CYP19A1CYP11B1CYP11B2
SCHEMBL22969568 0.66 GABRP (0.37) HTR2ASRD5A1CYP19A1CYP11B1CYP11B2
SCHEMBL8919270 0.65 NPC1 (0.47) HTR2ASRD5A1CYP19A1CYP11B1CYP11B2
SCHEMBL16135231 0.63 CYP11B2 (0.51) SRD5A1CYP19A1CYP11B1CYP11B2NPC1
SCHEMBL10595981 0.62 SMN1; SMN2 (0.49) SRD5A1CYP19A1CYP11B1CYP11B2NPC1
SCHEMBL434004 0.61 NPC1 (0.50) SRD5A1CYP19A1CYP11B1CYP11B2NPC1
SCHEMBL12090742 0.61 CYP19A1 (0.48) CYP19A1CYP11B1CYP11B2NPC1MAPK13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0294647-B1 THIADIAZINONES MERCK PATENT GmbH (DE) 1993-07-21 EP disclosed