SCHEMBL9533304

SCHEMBL9533304

CN(C)C=C1C(=O)CCc2c1cnn2C

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.51
CSNK2A1 P68400 1/20 0.51
PLK3 Q9H4B4 1/20 0.51
ALDH1A1 P00352 4/20 0.34
SMN1; SMN2 Q16637 3/20 0.34
HIF1A Q16665 2/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34
MAP1LC3B Q9GZQ8 4/20 0.32
RECQL P46063 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
POLB P06746 1/20 0.31
HSD17B10 Q99714 1/20 0.30
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9533291 1.00 PLK1 (0.51) PLK1CSNK2A1PLK3ALDH1A1SMN1; SMN2
SCHEMBL9534422 0.91 PLK1 (0.65) PLK1CSNK2A1PLK3ALDH1A1SMN1; SMN2
SCHEMBL22980483 0.78 PLK1 (0.79) PLK1CSNK2A1PLK3ALDH1A1SMN1; SMN2
SCHEMBL9535703 0.72 PLK1 (0.61) PLK1CSNK2A1PLK3ALDH1A1SMN1; SMN2
Hydrochloric Acid SCHEMBL9534437 0.70 PLK1 (0.59) PLK1CSNK2A1PLK3ALDH1A1SMN1; SMN2
SCHEMBL6837311 0.70 MAP1LC3B (0.47) ALDH1A1SMN1; SMN2HIF1AMAPTHTT
SCHEMBL3142557 0.68 PLK1 (0.93) PLK1CSNK2A1PLK3ALDH1A1SMN1; SMN2
SCHEMBL1986758 0.68 PLK1 (1.00) PLK1CSNK2A1PLK3ALDH1A1SMN1; SMN2
SCHEMBL9211876 0.66 PLK1 (0.50) PLK1CSNK2A1PLK3ALDH1A1SMN1; SMN2
SCHEMBL9211872 0.66 PLK1 (0.50) PLK1CSNK2A1PLK3ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276834-B1 Cycloalkane [1,2-c:4,3-c'] dipyrazoles MERRELL DOW PHARMACEUTICALS INC. (US) 1993-06-02 EP disclosed
EP-0525129-A4 SUBSTITUTED BENZIMIDAZOLES 1993-03-24 EP disclosed
EP-0525129-A1 SUBSTITUTED BENZIMIDAZOLES SMITHKLINE BEECHAM CORPORATION (US) 1993-02-03 EP disclosed
EP-0276834-A1 Cycloalkane [1,2-c:4,3-c'] dipyrazoles MERRELL DOW PHARMACEUTICALS INC. (US) 1988-08-03 EP disclosed
US-4734429-A Cycloalkane[1,2-c:4,3-c']dipyrazoles and their use as bronchodilators MERRELL DOW PHARMACEUTICALS INC. (US) 1988-03-29 US disclosed