SCHEMBL9534422

SCHEMBL9534422

CN(C)C=C1C(=O)CCCc2c1cnn2C

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PLK1 P53350 1/20 0.65
CSNK2A1 P68400 1/20 0.65
PLK3 Q9H4B4 1/20 0.65
HTT P42858 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
POLB P06746 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
TP53 P04637 1/20 0.37
CTDSP1 Q9GZU7 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
ELANE P08246 2/20 0.37
ALDH1A1 P00352 2/20 0.35
CYP11B2 P19099 2/20 0.34
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
CA4 P22748 2/20 0.33
CA9 Q16790 2/20 0.33
HIF1A Q16665 2/20 0.33
MAPT P10636 2/20 0.33
HTR1A P08908 3/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9533291 0.91 PLK1 (0.51) PLK1CSNK2A1PLK3HTTSMN1; SMN2
SCHEMBL9533304 0.91 PLK1 (0.51) PLK1CSNK2A1PLK3HTTSMN1; SMN2
SCHEMBL1986758 0.80 PLK1 (1.00) PLK1CSNK2A1PLK3HTTSMN1; SMN2
SCHEMBL3142557 0.76 PLK1 (0.93) PLK1CSNK2A1PLK3HTTSMN1; SMN2
SCHEMBL9533936 0.74 PLK1 (0.74) PLK1CSNK2A1PLK3HTTSMN1; SMN2
SCHEMBL955853 0.72 SMN1; SMN2 (0.57) HTTSMN1; SMN2POLBL3MBTL1TP53
SCHEMBL9535827 0.71 HTT (0.43) PLK1CSNK2A1PLK3HTTSMN1; SMN2
SCHEMBL22980483 0.69 PLK1 (0.79) PLK1CSNK2A1PLK3HTTSMN1; SMN2
SCHEMBL3142596 0.68 SMN1; SMN2 (0.52) HTTSMN1; SMN2POLBL3MBTL1TP53
SCHEMBL9214131 0.68 PLK1 (0.59) PLK1CSNK2A1PLK3HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276834-B1 Cycloalkane [1,2-c:4,3-c'] dipyrazoles MERRELL DOW PHARMACEUTICALS INC. (US) 1993-06-02 EP disclosed
EP-0276834-A1 Cycloalkane [1,2-c:4,3-c'] dipyrazoles MERRELL DOW PHARMACEUTICALS INC. (US) 1988-08-03 EP disclosed
US-4734429-A Cycloalkane[1,2-c:4,3-c']dipyrazoles and their use as bronchodilators MERRELL DOW PHARMACEUTICALS INC. (US) 1988-03-29 US disclosed