SCHEMBL9533760

SCHEMBL9533760

Cn1nc2ccc3nc(O)c(O)nc3c2n1

nearest known ligand 0.31

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.31
MAPT P10636 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9532966 0.73 SLC9A1 (0.39) KDM4EMAPT
SCHEMBL9533409 0.71 MAPT (0.50) KDM4EMAPTMAPK1
SCHEMBL9532647 0.69 ADRA2A (0.37) KDM4EMAPTMAPK1
SCHEMBL9496336 0.68 F2 (0.40) MAPTMAPK1
SCHEMBL9532856 0.67 DPP4 (0.38) KDM4E
SCHEMBL822536 0.65 SLC2A1 (0.58) KDM4EMAPTMAPK1
SCHEMBL5984487 0.64 ACHE (0.39) KDM4EMAPTMAPK1
SCHEMBL24402911 0.64 CCR1 (0.35) MAPTMAPK1
SCHEMBL9534598 0.64 MAPT (0.41) KDM4EMAPTMAPK1
SCHEMBL9534618 0.64 POLB (0.42) KDM4EMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4977155-A Nervous system disorders A/S FERROSAN (DK) 1990-12-11 US claimed
EP-0348872-B1 FUSED DIHYDROXYQUINOXALINES AND THEIR USE AS GLUTAMATE ANTAGONISTS NOVO NORDISK A/S (DK) 1993-09-29 EP disclosed
US-5109001-A Treating hyperactivity of excitatory neurotransmitters NOVO NORDISK A/S (DK) 1992-04-28 US disclosed
US-5079250-A TRICYCLIC HETEROCYCLIC DIOLS AND THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 1992-01-07 US disclosed
US-5075306-A Nervous system, psychological disorders NOVO NORDISK A/S (DK) 1991-12-24 US disclosed
US-5057516-A Nervous system disorders NOVO NORDISK A/S (DK) 1991-10-15 US disclosed
US-4977155-A Nervous system disorders A/S FERROSAN (DK) 1990-12-11 US disclosed
EP-0348872-A1 Fused dihydroxyquinoxalines and their use as glutamate antagonists NOVO NORDISK A/S (DK) 1990-01-03 EP disclosed