SCHEMBL9534217

SCHEMBL9534217

Cc1onc(-c2c(F)cccc2Cl)c1OC(=O)Nc1ccc(SC(F)(F)F)cc1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.51
MAPT P10636 1/20 0.51
PTGS2 P35354 5/20 0.51
LMNA P02545 3/20 0.51
GLA P06280 2/20 0.51
ATM Q13315 2/20 0.51
HPGD P15428 1/20 0.51
HTT P42858 1/20 0.51
SCN9A Q15858 2/20 0.49
PRNP P04156 1/20 0.47
RXFP1 Q9HBX9 1/20 0.47
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
ALDH1A1 P00352 2/20 0.46
SCN5A Q14524 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9536336 0.80 SCN9A (0.54) TP53MAPTLMNAGLAATM
SCHEMBL9536259 0.78 PTGS2 (0.50) TP53MAPTPTGS2LMNAGLA
SCHEMBL9536365 0.77 LMNA (0.57) TP53MAPTLMNAGLAATM
SCHEMBL5242736 0.77 ALDH1A1 (0.58) LMNAGLAATMHPGDHTT
SCHEMBL9537042 0.72 SMN1; SMN2 (0.54) TP53MAPTLMNAGLAATM
SCHEMBL9537606 0.71 KDM4E (0.50) TP53MAPTLMNAGLAATM
SCHEMBL9535763 0.71 KMT2A (0.58) PTGS2LMNAGLAATMHPGD
SCHEMBL9535614 0.70 TSHR (0.53) MAPTPTGS2LMNAGLAHPGD
SCHEMBL12584906 0.70 SCN9A (0.67) TP53MAPTLMNAGLAATM
SCHEMBL11893412 0.69 ALDH1A1 (0.72) TP53MAPTLMNAGLAATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0573883-A1 Utilization of 3 substituted aryl-5-alkyl-isoxazole-4-carboxylic acid derivatives against endoparasites new 3-substituted aryl-5-alkyl-isoxazole-4-carboxylic acid derivatives and process for their preparation BAYER AG (DE) 1993-12-15 EP disclosed