SCHEMBL9534341

SCHEMBL9534341

CCn1cc(C(=O)O)c(=O)c2cc(F)c(N3CC4=C(C3)C(N)CC4)c(F)c21

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.58
ALDH1A1 P00352 5/20 0.58
HSD17B10 Q99714 4/20 0.58
HPGD P15428 4/20 0.58
PMP22 Q01453 1/20 0.57
KCNH2 Q12809 3/20 0.43
DRD3 P35462 1/20 0.43
LMNA P02545 3/20 0.42
BRD4 O60885 1/20 0.42
TSHR P16473 1/20 0.42
HTT P42858 1/20 0.42
CYP2J2 P51589 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
TOP1 P11387 2/20 0.42
POLB P06746 1/20 0.41
CHRM2 P08172 1/20 0.41
CHRM1 P11229 1/20 0.41
OPRM1 P35372 1/20 0.41
OPRD1 P41143 1/20 0.41
CYP2C9 P11712 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9241429 0.86 ALDH1A1 (0.54) KDM4EALDH1A1HSD17B10HPGDKCNH2
SCHEMBL9536182 0.85 KDM4E (0.43) KDM4EALDH1A1HSD17B10HPGDPMP22
SCHEMBL9534442 0.84 DRD3 (0.61) KDM4EALDH1A1HSD17B10HPGDDRD3
SCHEMBL9537372 0.84 CACNA1F (0.47) KDM4EALDH1A1HSD17B10HPGDPMP22
SCHEMBL9537286 0.83 KDM4E (0.46) KDM4EALDH1A1HSD17B10HPGDLMNA
SCHEMBL9535029 0.82 LMNA (0.61) KDM4EALDH1A1HSD17B10HPGDDRD3
SCHEMBL9535373 0.82 KMT2A (0.49) KDM4EALDH1A1HSD17B10HPGDLMNA
SCHEMBL8699900 0.80 ALDH1A1 (0.71) KDM4EALDH1A1HSD17B10HPGDPMP22
SCHEMBL9535876 0.80 KDM4E (0.48) KDM4EALDH1A1HSD17B10HPGDPMP22
SCHEMBL9535599 0.80 ALDH1A1 (0.49) KDM4EALDH1A1HSD17B10HPGDKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993013090-A1 NOVEL QUINOLONE CARBOXYLIC ACID DERIVATIVES AND PROCESSES FOR PREPARING SAME HOECHST AKTIENGESELLSCHAFT (DE) 1993-07-08 WO disclosed
EP-0549857-A1 Antibacterial quinolone carboxylic acid derivatives KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 1993-07-07 EP disclosed