SCHEMBL9535827

SCHEMBL9535827

Cc1nn(C)c2c1C(=CN(C)C)C(=O)CCC2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.37
TP53 P04637 1/20 0.37
POLB P06746 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CTDSP1 Q9GZU7 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
ALOX15 P16050 1/20 0.36
CYP2C19 P33261 1/20 0.36
CREBBP Q92793 1/20 0.36
HSD17B10 Q99714 1/20 0.36
PLK1 P53350 1/20 0.36
CSNK2A1 P68400 1/20 0.36
PLK3 Q9H4B4 1/20 0.36
OPRM1 P35372 1/20 0.35
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6164696 0.80 HTT (0.61) HTTLMNAMAPTPLK1CSNK2A1
SCHEMBL955853 0.72 SMN1; SMN2 (0.57) HTTL3MBTL1TP53POLBSMN1; SMN2
SCHEMBL9534422 0.71 PLK1 (0.65) HTTL3MBTL1TP53POLBSMN1; SMN2
SCHEMBL3142596 0.68 SMN1; SMN2 (0.52) HTTL3MBTL1TP53POLBSMN1; SMN2
SCHEMBL21635879 0.66 SMN1; SMN2 (0.50) HTTL3MBTL1TP53POLBSMN1; SMN2
SCHEMBL21678821 0.65 HTT (0.38) HTTPARP1
SCHEMBL6837311 0.64 MAP1LC3B (0.47) HTTL3MBTL1TP53POLBSMN1; SMN2
SCHEMBL6166619 0.63 HTT (0.42) HTTLMNAPLK1CSNK2A1PLK3
SCHEMBL9533291 0.62 PLK1 (0.51) HTTL3MBTL1POLBSMN1; SMN2MAPT
SCHEMBL9533304 0.62 PLK1 (0.51) HTTL3MBTL1POLBSMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0276834-B1 Cycloalkane [1,2-c:4,3-c'] dipyrazoles MERRELL DOW PHARMACEUTICALS INC. (US) 1993-06-02 EP disclosed
EP-0276834-A1 Cycloalkane [1,2-c:4,3-c'] dipyrazoles MERRELL DOW PHARMACEUTICALS INC. (US) 1988-08-03 EP disclosed
US-4734429-A Cycloalkane[1,2-c:4,3-c']dipyrazoles and their use as bronchodilators MERRELL DOW PHARMACEUTICALS INC. (US) 1988-03-29 US disclosed