SCHEMBL9534817

SCHEMBL9534817

O=C(O)Cc1ccc(-c2cc3ccccc3c3ccccc23)[nH]c1=O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.45
AKR1B1 P15121 2/20 0.42
DHODH Q02127 1/20 0.41
LCK P06239 1/20 0.39
PRKACA P17612 1/20 0.39
CSNK2A2 P19784 1/20 0.39
PRKACG P22612 1/20 0.39
PRKACB P22694 1/20 0.39
GSK3B P49841 1/20 0.39
CSNK2B P67870 1/20 0.39
CSNK2A1 P68400 1/20 0.39
DYRK1A Q13627 1/20 0.39
CSNK2A3 Q8NEV1 1/20 0.39
KDM4E B2RXH2 4/20 0.39
ALDH1A1 P00352 3/20 0.39
GAA P10253 2/20 0.39
GLA P06280 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
MAPT P10636 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9538652 0.85 TDP1 (0.54) TDP1AKR1B1LCKPRKACACSNK2A2
SCHEMBL9754429 0.79 KDM4E (0.58) KDM4EALDH1A1GAAGLAHPGD
SCHEMBL9534054 0.77 PTGER3 (0.53) KDM4EALDH1A1HPGDHSD17B10CYP1A2
SCHEMBL9539842 0.75 KDM4E (0.42) KDM4EALDH1A1GAAHPGDHSD17B10
SCHEMBL9535637 0.75 PTGER3 (0.39) AKR1B1DHODHKDM4EALDH1A1GAA
SCHEMBL9095402 0.74 CHEK1 (0.48) TDP1AKR1B1KDM4EALDH1A1GAA
SCHEMBL9536127 0.72 KDM4E (0.37) KDM4EALDH1A1GAAHPGDMAPT
SCHEMBL9536884 0.70 KDM4E (0.46) DYRK1AKDM4EALDH1A1GAAGLA
SCHEMBL11665605 0.70 LOXL2 (0.62) TDP1AKR1B1LCKPRKACACSNK2A2
SCHEMBL9536629 0.69 APAF1 (0.40) KDM4EALDH1A1GAAGLAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991017987-A1 PHENOL AND PYRIDINOL DERIVATIVES AS PHARMACEUTICALS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1991-11-28 WO claimed
EP-0532531-A1 PHENOL AND PYRIDINOL DERIVATIVES AS PHARMACEUTICALS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1993-03-24 EP disclosed
WO-1991017987-A1 PHENOL AND PYRIDINOL DERIVATIVES AS PHARMACEUTICALS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1991-11-28 WO disclosed