SCHEMBL9534906

SCHEMBL9534906

c1ccc(CN2CCC(Cc3nc4cnccc4[nH]3)CC2)cc1

nearest known ligand 0.64

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GRIN2B Q13224 7/20 0.64
GRIN1 Q05586 5/20 0.64
HRH3 Q9Y5N1 2/20 0.54
CCR3 P51677 1/20 0.53
ALDH1A1 P00352 2/20 0.48
ROCK2 O75116 1/20 0.46
ROCK1 Q13464 1/20 0.46
KDM4E B2RXH2 1/20 0.45
GLA P06280 1/20 0.45
GAA P10253 1/20 0.45
MAPT P10636 1/20 0.45
HTT P42858 1/20 0.45
ATM Q13315 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
IDO1 P14902 1/20 0.45
HTR2B P41595 2/20 0.45
GRIN2A Q12879 1/20 0.45
DRD4 P21917 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7012695 0.92 GRIN2B (0.77) GRIN2BGRIN1HRH3CCR3ALDH1A1
SCHEMBL7972912 0.87 GRIN2B (0.83) GRIN2BGRIN1HRH3CCR3ALDH1A1
SCHEMBL9537890 0.81 GRIN2B (0.63) GRIN2BGRIN1HRH3CCR3ALDH1A1
SCHEMBL1388535 0.78 GRIN2B (1.00) GRIN2BGRIN1CCR3HTTIDO1
SCHEMBL8628385 0.77 AAK1 (0.59) GRIN2BGRIN1IDO1
SCHEMBL10548102 0.76 THRB (0.64) GRIN2BGRIN1DRD4
SCHEMBL7073777 0.76 GRIN2B (0.52) GRIN2BGRIN1ROCK2ROCK1IDO1
SCHEMBL10552369 0.74 THRB (0.59) GRIN2BGRIN1CCR3DRD4
SCHEMBL5237195 0.73 GRIN1 (0.84) GRIN2BGRIN1CCR3GAAGRIN2A
SCHEMBL7241045 0.73 GRIN1 (0.65) GRIN2BGRIN1HRH3CCR3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP disclosed
US-4839374-A TREATING ALLERGIES JANSSEN PHARMACEUTICA, N.V. (BE) 1989-06-13 US disclosed
US-4695575-A ANTIHISTAMINES JANSSEN PHARMACEUTICA, N.V. (BE) 1987-09-22 US disclosed