SCHEMBL9535982

SCHEMBL9535982

CCOC(=O)c1nnsc1-c1ccc([O])cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2C9 P11712 1/20 0.51
HSD17B10 Q99714 1/20 0.51
MAPT P10636 4/20 0.50
MEN1 O00255 2/20 0.50
KMT2A Q03164 2/20 0.50
ILK Q13418 1/20 0.50
HTT P42858 1/20 0.50
TSHR P16473 1/20 0.49
KDM4E B2RXH2 1/20 0.44
POLB P06746 1/20 0.44
TARBP2 Q15633 5/20 0.41
NPSR1 Q6W5P4 1/20 0.39
GRM6 O15303 2/20 0.39
PDCD4 Q53EL6 1/20 0.39
TP53 P04637 1/20 0.38
ALOX12 P18054 1/20 0.38
LMNA P02545 1/20 0.38
PKM P14618 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9535985 0.89 ALDH1A1 (0.51) ALDH1A1CYP1A2CYP2C9HSD17B10MAPT
SCHEMBL22230643 0.87 TARBP2 (0.53) ALDH1A1CYP1A2CYP2C9HSD17B10MAPT
SCHEMBL6815148 0.87 ILK (0.61) ALDH1A1CYP1A2CYP2C9HSD17B10MAPT
SCHEMBL11773257 0.79 ILK (0.49) ALDH1A1HSD17B10MAPTMEN1KMT2A
SCHEMBL7586906 0.78 ILK (0.55) ALDH1A1CYP1A2CYP2C9HSD17B10MAPT
SCHEMBL9536015 0.77 ALDH1A1 (0.43) ALDH1A1CYP1A2CYP2C9HSD17B10MAPT
SCHEMBL11771172 0.75 ILK (0.54) ALDH1A1HSD17B10MAPTMEN1KMT2A
SCHEMBL11770705 0.74 ADRB2 (0.48) CYP1A2MAPTMEN1KMT2ATSHR
SCHEMBL11773521 0.73 ADRB2 (0.49) MAPTMEN1KMT2AHTT
SCHEMBL7794327 0.73 TSHR (0.61) ALDH1A1CYP1A2MAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0375560-B1 ARYLOXYPROPANOLAMINOTETRALINES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING SAME ELF SANOFI (FR) 1993-05-12 EP disclosed