SCHEMBL9536636

SCHEMBL9536636

O=C(NCCCCN1CCC(Cc2nc3ccccc3n2Cc2ccc(F)cc2)CC1)c1ccccc1

nearest known ligand 0.65

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR3 P51677 6/20 0.65
TMEM97 Q5BJF2 4/20 0.55
MAPT P10636 1/20 0.54
TP53 P04637 2/20 0.51
POLB P06746 2/20 0.50
SLC6A2 P23975 1/20 0.50
SLC6A4 P31645 1/20 0.50
KCNH2 Q12809 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9536186 0.94 MAPT (0.56) CCR3MAPTTP53POLBSLC6A2
SCHEMBL10549253 0.89 CCR3 (0.52) CCR3TMEM97POLBKCNH2
SCHEMBL9536165 0.85 CCR3 (0.56) CCR3TMEM97MAPTPOLBSLC6A2
Oxalic Acid SCHEMBL9538011 0.84 PLD2 (0.47) CCR3MAPTTP53POLBSLC6A2
Oxalic Acid SCHEMBL9538009 0.84 PLD2 (0.47) CCR3MAPTTP53POLBSLC6A2
SCHEMBL9536847 0.84 KCNH2 (0.49) TP53POLBKCNH2
Oxalic Acid SCHEMBL10552513 0.83 SSTR5 (0.51) TP53KCNH2
SCHEMBL10547215 0.83 POLB (0.49) CCR3POLBSLC6A2SLC6A4KCNH2
SCHEMBL9536213 0.83 TP53 (0.61) CCR3MAPTTP53POLB
SCHEMBL9539669 0.82 RAB9A (0.52) TMEM97MAPTTP53SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP disclosed