SCHEMBL9537387

SCHEMBL9537387

C=C(c1cccnc1)c1ncc(O)c(C(C)(C)C)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.38
LMNA P02545 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP11B1 P15538 1/20 0.38
CYP11B2 P19099 1/20 0.38
ALDH1A1 P00352 3/20 0.36
THRB P10828 1/20 0.36
APP P05067 2/20 0.36
GSK3B P49841 1/20 0.36
ESR1 P03372 1/20 0.35
GAA P10253 1/20 0.35
HCAR3 P49019 1/20 0.35
HCAR2 Q8TDS4 1/20 0.35
RAB9A P51151 1/20 0.34
F7 P08709 1/20 0.34
F3 P13726 1/20 0.34
SARM1 Q6SZW1 1/20 0.34
SIRT2 Q8IXJ6 1/20 0.34
SIRT6 Q8N6T7 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9301523 0.85 TDP1 (0.40) TDP1LMNACYP1A2CYP3A4CYP11B1
SCHEMBL9539358 0.74 CYP3A4 (0.48) TDP1LMNACYP1A2CYP3A4ALDH1A1
SCHEMBL8865984 0.70 ALDH1A1 (0.58) TDP1LMNACYP1A2CYP3A4CYP11B1
SCHEMBL9537381 0.68 ALOX5 (0.53) CYP1A2CYP11B1CYP11B2RAB9ASMN1; SMN2
SCHEMBL9304107 0.67 KMT2A (0.37) TDP1LMNAALDH1A1RAB9ASMN1; SMN2
SCHEMBL800783 0.67 LMNA (0.51) TDP1LMNACYP1A2CYP3A4CYP11B1
SCHEMBL9431575 0.66 GLRA3 (0.32)
SCHEMBL9405525 0.65 BAZ2B (0.31)
SCHEMBL29721526 0.65 ALDH1A1 (0.57) TDP1LMNACYP1A2CYP3A4CYP11B1
SCHEMBL9412699 0.65 ALDH1A1 (0.57) TDP1LMNACYP1A2CYP3A4CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0569491-A4 2-SUBSTITUTED-4,6-DI-TERTIARY-BUTYL-5-HYDROXY-1,3-PYRIMIDINES USEFUL AS ANTIINFLAMMATORY AGENTS 1993-11-24 EP claimed