SCHEMBL9537953

SCHEMBL9537953

Cc1nc2ccccn2c(=O)c1CCN1CCC(Cc2nc3cccnc3n2Cc2ccco2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.46
MAPT P10636 5/20 0.46
MEN1 O00255 4/20 0.46
KMT2A Q03164 4/20 0.46
HPGD P15428 3/20 0.46
HTR1A P08908 2/20 0.46
HTR2C P28335 2/20 0.46
PKM P14618 2/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2D6 P10635 1/20 0.46
TSHR P16473 1/20 0.46
THPO P40225 1/20 0.46
PMP22 Q01453 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
ACHE P22303 1/20 0.42
ADRA1A P35348 5/20 0.41
ADRA2A P08913 5/20 0.41
ADRA2B P18089 5/20 0.41
ADRA2C P18825 5/20 0.41
DRD2 P14416 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9536415 0.90 KDM4E (0.48) KDM4EMAPTMEN1KMT2AHPGD
SCHEMBL9538894 0.87 SLC6A9 (0.44) KDM4EMAPTMEN1KMT2AHPGD
Barmastine SCHEMBL141926 0.86 KDM4E (0.45) KDM4EMAPTMEN1KMT2AHPGD
Barmastine SCHEMBL30712053 0.86 KDM4E (0.45) KDM4EMAPTMEN1KMT2AHPGD
SCHEMBL9537351 0.86 HTR1A (0.56) KDM4EMAPTMEN1KMT2AHPGD
SCHEMBL9535132 0.84 SLC6A9 (0.43) MAPTHTR1ATSHRDRD2HTR2A
SCHEMBL9536136 0.83 SLC6A9 (0.44) KDM4EHPGDHTR1ATSHRDRD2
Hydrochloric Acid SCHEMBL9535191 0.82 SLC6A9 (0.43) KDM4EHPGDHTR1ATSHRDRD2
SCHEMBL9538129 0.80 GAA (0.51) KDM4EMAPTHTR1ATSHRSMN1; SMN2
SCHEMBL9537181 0.78 SLC6A9 (0.49) KDM4EMAPTMEN1KMT2AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP claimed