SCHEMBL9536136

SCHEMBL9536136

Cc1nc2scc(C)n2c(=O)c1CCN1CCC(Cc2nc3cccnc3n2Cc2ccco2)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 1/20 0.44
LMNA P02545 1/20 0.36
ALDH1A1 P00352 4/20 0.35
HPGD P15428 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
KDM4E B2RXH2 1/20 0.35
RECQL P46063 1/20 0.35
HSD17B10 Q99714 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ADORA2A P29274 2/20 0.34
ADORA2B P29275 2/20 0.34
MAPK1 P28482 2/20 0.34
GAA P10253 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
HTT P42858 1/20 0.33
POLB P06746 3/20 0.33
TSHR P16473 4/20 0.33
BRD4 O60885 1/20 0.32
BRD2 P25440 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9535191 0.99 SLC6A9 (0.43) SLC6A9LMNAALDH1A1HPGDTDP1
SCHEMBL9536406 0.89 ALDH1A1 (0.37) ALDH1A1HPGDTDP1KDM4ERECQL
SCHEMBL9538894 0.88 SLC6A9 (0.44) SLC6A9LMNAALDH1A1HPGDTDP1
SCHEMBL9535132 0.84 SLC6A9 (0.43) SLC6A9LMNAALDH1A1HSD17B10ADORA2A
SCHEMBL9537953 0.83 KDM4E (0.46) SLC6A9LMNAALDH1A1HPGDTDP1
SCHEMBL9538129 0.77 GAA (0.51) SLC6A9LMNAALDH1A1TDP1KDM4E
SCHEMBL9537181 0.77 SLC6A9 (0.49) SLC6A9LMNAALDH1A1HPGDTDP1
SCHEMBL9535079 0.77 TSHR (0.45) LMNAALDH1A1HPGDTDP1KDM4E
SCHEMBL9564914 0.76 CYP3A4 (0.47) SLC6A9LMNAALDH1A1HPGDTDP1
SCHEMBL9536805 0.75 SLC6A9 (0.51) SLC6A9LMNAALDH1A1HPGDTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP claimed