SCHEMBL9538129

SCHEMBL9538129

Cc1nc2ccccc2c(=O)n1CCN1CCC(Cc2nc3cccnc3n2Cc2ccco2)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.51
TSHR P16473 9/20 0.46
ALDH1A1 P00352 8/20 0.46
MAPK1 P28482 3/20 0.45
NPSR1 Q6W5P4 3/20 0.45
SLC6A9 P48067 1/20 0.45
HTT P42858 2/20 0.44
LMNA P02545 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
HSD17B10 Q99714 2/20 0.41
ALOX15 P16050 1/20 0.41
HTR1A P08908 1/20 0.41
HTR7 P34969 1/20 0.41
USP2 O75604 2/20 0.41
CACNA2D1 P54289 1/20 0.41
HIF1A Q16665 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
POLB P06746 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9537429 0.89 GAA (0.52) GAATSHRALDH1A1MAPK1NPSR1
SCHEMBL9535214 0.86 SLC6A9 (0.41) GAATSHRALDH1A1MAPK1NPSR1
SCHEMBL9540573 0.85 SLC6A9 (0.52) GAAALDH1A1SLC6A9LMNAHTR1A
SCHEMBL9539651 0.85 ALDH1A1 (0.47) TSHRALDH1A1SMN1; SMN2HSD17B10ALOX15
SCHEMBL9537181 0.82 SLC6A9 (0.49) GAATSHRALDH1A1MAPK1NPSR1
SCHEMBL9537207 0.82 SLC6A9 (0.47) TSHRALDH1A1MAPK1NPSR1SLC6A9
Water SCHEMBL10554595 0.82 SLC6A9 (0.41) GAATSHRALDH1A1MAPK1NPSR1
SCHEMBL9540587 0.82 TSHR (0.50) GAATSHRALDH1A1MAPK1NPSR1
SCHEMBL10550979 0.82 TSHR (0.50) GAATSHRALDH1A1MAPK1NPSR1
SCHEMBL10549053 0.81 HSD17B10 (0.42) GAATSHRALDH1A1MAPK1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP disclosed
US-4839374-A TREATING ALLERGIES JANSSEN PHARMACEUTICA, N.V. (BE) 1989-06-13 US disclosed
US-4695575-A ANTIHISTAMINES JANSSEN PHARMACEUTICA, N.V. (BE) 1987-09-22 US disclosed