SCHEMBL9537207

SCHEMBL9537207

c1ccc(CN2CCC(Cc3nc4cccnc4n3Cc3ccco3)CC2)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 1/20 0.47
ALDH1A1 P00352 3/20 0.45
POLB P06746 1/20 0.45
HPGD P15428 1/20 0.45
TSHR P16473 1/20 0.45
MAPK1 P28482 1/20 0.45
HSD17B10 Q99714 1/20 0.45
LMNA P02545 3/20 0.44
CCR3 P51677 1/20 0.44
ENPP2 Q13822 3/20 0.44
TP53 P04637 1/20 0.42
HTR3E A5X5Y0 1/20 0.41
HTR3B O95264 1/20 0.41
HTR1A P08908 1/20 0.41
HTR2C P28335 1/20 0.41
HTR3A P46098 1/20 0.41
HTR3D Q70Z44 1/20 0.41
HTR3C Q8WXA8 1/20 0.41
ACHE P22303 1/20 0.41
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9537927 0.89 LMNA (0.55) SLC6A9ALDH1A1LMNACCR3ENPP2
SCHEMBL9537181 0.86 SLC6A9 (0.49) SLC6A9ALDH1A1POLBHPGDTSHR
SCHEMBL9539854 0.86 ALDH1A1 (0.52) ALDH1A1TSHRHSD17B10LMNACCR3
SCHEMBL9536805 0.84 SLC6A9 (0.51) SLC6A9ALDH1A1POLBHPGDTSHR
SCHEMBL9535787 0.84 KDM4E (0.55) SLC6A9ALDH1A1LMNACCR3ENPP2
SCHEMBL9536624 0.83 SLC6A9 (0.47) SLC6A9ALDH1A1POLBHPGDTSHR
SCHEMBL9535367 0.83 SLC6A9 (0.58) SLC6A9LMNACCR3ENPP2TP53
SCHEMBL9536863 0.83 TP53 (0.54) SLC6A9ALDH1A1POLBLMNACCR3
SCHEMBL9537090 0.83 TP53 (0.44) SLC6A9ALDH1A1POLBHPGDTSHR
SCHEMBL9536027 0.83 SLC6A9 (0.67) SLC6A9POLBLMNACCR3ENPP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP disclosed
US-4839374-A TREATING ALLERGIES JANSSEN PHARMACEUTICA, N.V. (BE) 1989-06-13 US disclosed
US-4695575-A ANTIHISTAMINES JANSSEN PHARMACEUTICA, N.V. (BE) 1987-09-22 US disclosed
EP-0151826-A1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1985-08-21 EP disclosed