SCHEMBL9538832

SCHEMBL9538832

COc1ccc(Cc2ccc(F)cc2)c(N)c1N

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.43
HTT P42858 2/20 0.40
ALDH1A1 P00352 2/20 0.40
MAPT P10636 1/20 0.40
TSHR P16473 1/20 0.40
MAPK1 P28482 1/20 0.40
CA2 P00918 1/20 0.39
LTA4H P09960 1/20 0.39
KMT2A Q03164 2/20 0.38
DHFR P00374 1/20 0.38
POLB P06746 1/20 0.38
HPGD P15428 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
KDM4E B2RXH2 1/20 0.38
GPR55 Q9Y2T6 1/20 0.38
CYP17A1 P05093 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3788490 0.86 GAA (0.40) GAAHTTALDH1A1MAPTTSHR
SCHEMBL3038603 0.79 GAA (0.69) GAAHTTALDH1A1MAPTTSHR
SCHEMBL15906106 0.76 SMN1; SMN2 (0.41) GAAMAPTTSHRMAPK1LTA4H
SCHEMBL9535895 0.75 CNR1 (0.41) GAAALDH1A1SMN1; SMN2GPR55
SCHEMBL9538789 0.75 ALDH1A1 (0.46) GAAALDH1A1CA2KMT2APOLB
SCHEMBL3153666 0.75 KMT2A (0.56) GAAALDH1A1MAPTMAPK1LTA4H
SCHEMBL7859778 0.73 MAOB (0.42) GAAHTTMAPTTSHRMAPK1
SCHEMBL8070659 0.73 STK10 (0.38) GAAALDH1A1MAPTKMT2ASMN1; SMN2
SCHEMBL16158923 0.73 HTR1A (0.37) GAAALDH1A1LTA4HKMT2APOLB
SCHEMBL28846076 0.72 HTR1A (0.51) LTA4HHPGDSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP disclosed
EP-0151826-A1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1985-08-21 EP disclosed