SCHEMBL953930

SCHEMBL953930

CC(C(N)=O)c1cc(F)cc(-c2nnn[nH]2)c1

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.35
TRPM8 Q7Z2W7 2/20 0.33
NR1I2 O75469 1/20 0.33
SLC9A1 P19634 1/20 0.32
EPHX1 P07099 1/20 0.31
CTSA P10619 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL949480 0.82 CTSA (0.30) CTSA
SCHEMBL949999 0.80 APP (0.36) APPEPHX1CTSA
SCHEMBL953932 0.71 CAPN1 (0.34)
SCHEMBL17335564 0.70 PARP1 (0.34) CTSA
SCHEMBL949482 0.69 MPO (0.36)
SCHEMBL953933 0.68 CYP3A4 (0.40)
SCHEMBL17335530 0.67 APP (0.36) APP
SCHEMBL7383797 0.66 SLC9A1 (0.31) SLC9A1
SCHEMBL17335566 0.65 PARP1 (0.37) CTSA
SCHEMBL12479410 0.65 CASP1 (0.39)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011006935-A2 TETRAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2011-01-20 WO disclosed